Comparative biodistributions of yttrium- and indium-labeled monoclonal antibody B72.3 in athymic mice bearing human colon carcinoma xenografts

J Nucl Med. 1989 May;30(5):672-82.

Abstract

The biodistribution of yttrium- and indium-labeled monoclonal antibody (MAb) B72.3 IgG using three different chelate conjugates (SCN-Bz-EDTA, CA-DTPA, and SCN-Bz-DTPA) was compared in athymic mice bearing LS-174T tumors. The 88Y-SCN-Bz-DTPA-B72.3 yielded 40% ID/g at 5-7 days in the tumors, while the 88Y-SCN-Bz-EDTA-B72.3 and 88Y-CA-DTPA-B72.3 showed only 6-8% ID/g. The yttrium uptake in the bone with the SCN-Bz-EDTA and CA-DTPA conjugated IgG was over 14 and 11% ID/g, respectively, while 88Y-SCN-Bz-DTPA-B72.3 showed only 3% ID/g. In contrast, the 111In-labeled B72.3 uptake in the bone with all three chelate conjugates was 2-3% ID/g. The differences in yttrium- versus indium-labeled MAb biodistributions demonstrate the difficulty in using 111In-labeled MAbs to predict the biodistribution and dosimetry of 90Y-labeled MAbs unless chelate conjugates such as SCN-Bz-DTPA are used.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Antibodies, Monoclonal / metabolism*
  • Antibodies, Monoclonal / therapeutic use
  • Carcinoma / metabolism*
  • Carcinoma / radiotherapy
  • Chelating Agents / pharmacokinetics
  • Chelating Agents / therapeutic use
  • Colonic Neoplasms / metabolism*
  • Colonic Neoplasms / radiotherapy
  • Female
  • Humans
  • Immunoglobulin G / metabolism
  • Immunoglobulin G / therapeutic use
  • Immunotoxins / metabolism*
  • Immunotoxins / therapeutic use
  • Indium Radioisotopes / metabolism*
  • Indium Radioisotopes / therapeutic use
  • Mice
  • Mice, Nude / metabolism*
  • Neoplasm Transplantation
  • Tissue Distribution
  • Transplantation, Heterologous
  • Yttrium Radioisotopes / metabolism*
  • Yttrium Radioisotopes / therapeutic use

Substances

  • Antibodies, Monoclonal
  • Chelating Agents
  • Immunoglobulin G
  • Immunotoxins
  • Indium Radioisotopes
  • Yttrium Radioisotopes