Mesenchymal stromal cell-secreted chemerin is a novel immunomodulatory molecule driving the migration of ChemR23-expressing cells

Cytotherapy. 2017 Feb;19(2):200-210. doi: 10.1016/j.jcyt.2016.11.006. Epub 2016 Dec 6.

Abstract

Background: Mesenchymal stromal cells (MSCs) are multipotent cells characterized by broad immunomodulatory properties exploited for the treatment of inflammatory disorders. However, the efficacy of MSC-based therapy is highly variable and tightly linked to MSC culture conditions and treatment schedule. Thus, the identification of novel key molecules regulating MSC immunomodulatory activities in vivo might constitute a crucial step toward the optimization of currently available clinical protocols. In this regard, herein, we sought to determine whether the newly identified chemotactic protein, chemerin, plays a role in MSC-mediated regulation of inflammation.

Methods: Chemerin production by human MSCs was investigated under different culture conditions using enzyme-linked immunosorbent assay (ELISA). After purification, MSC-secreted chemerin was identified using mass spectrometry analysis and the biological activity of secreted isoforms was evaluated using migration assay.

Results: Bone marrow-derived MSCs secrete chemerin and express its receptors ChemR23 and CCRL2. Chemerin production is dependent on culture conditions and increases upon stimulation with inflammatory cytokines. In particular, platelet lysate (PL)-MSCs produce higher levels of chemerin compared with fetal bovine serum (FBS)-MSCs. Furthermore, chemerin is secreted by MSCs as an inactive precursor, which can be converted into its active form by exogenous chemerin-activating serine and cysteine proteases.

Discussion: Our data indicate that, in response to various inflammatory stimuli, MSCs secrete high amounts of inactive chemerin, which can then be activated by inflammation-induced tissue proteases. In light of these initial findings, we propose that further analysis of chemerin functions in vivo might constitute a crucial step toward optimizing MSC-based therapy for inflammatory diseases.

Keywords: ChemR23 receptor; chemerin; immunomodulation; mesenchymal stromal cells.

MeSH terms

  • Blood Platelets / chemistry
  • Cell Culture Techniques
  • Cell Extracts / chemistry
  • Cell Extracts / pharmacology
  • Cells, Cultured
  • Chemotaxis / drug effects*
  • Chemotaxis / genetics
  • Chimerin Proteins / genetics
  • Chimerin Proteins / metabolism
  • Chimerin Proteins / pharmacology*
  • Culture Media / metabolism
  • Culture Media / pharmacology
  • Human Umbilical Vein Endothelial Cells
  • Humans
  • Immunomodulation / drug effects*
  • Immunomodulation / genetics
  • Inflammation / metabolism
  • Inflammation / therapy
  • Mesenchymal Stem Cell Transplantation / methods
  • Mesenchymal Stem Cells / cytology
  • Mesenchymal Stem Cells / metabolism*
  • Receptors, Chemokine / genetics
  • Receptors, Chemokine / metabolism*

Substances

  • CMKLR1 protein, human
  • Cell Extracts
  • Chimerin Proteins
  • Culture Media
  • Receptors, Chemokine