Nudix-type motif 2 contributes to cancer proliferation through the regulation of Rag GTPase-mediated mammalian target of rapamycin complex 1 localization

Cell Signal. 2017 Apr:32:24-35. doi: 10.1016/j.cellsig.2017.01.015. Epub 2017 Jan 13.

Abstract

Lysosomal localization of mammalian target of rapamycin complex 1 (mTORC1) is a critical step for activation of the molecule. Rag GTPases are essential for this translocation. Here, we demonstrate that Nudix-type motif 2 (NUDT2) is a novel positive regulator of mTORC1 activation. Activation of mTORC1 is impaired in NUDT2-silenced cells. Mechanistically, NUDT2 binds to Rag GTPase and controls mTORC1 translocation to the lysosomal membrane. Furthermore, NUDT2-dependent mTORC1 regulation is critical for proliferation of breast cancer cells, as NUDT2-silenced cells arrest in G0/G1 phases. Taken together, these results show that NUDT2 is a novel complex formation enhancing factor regulating mTORC1-Rag GTPase signaling that is crucial for cell growth control.

Keywords: Cancer cell proliferation; Lysosomal localization; Mammalian target of rapamycin complex 1 (mTORC1); Nudix-type motif 2 (NUDT2); Rag GTPases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acids / pharmacology
  • Cell Cycle Checkpoints / drug effects
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • G1 Phase / drug effects
  • Gene Knockdown Techniques
  • Humans
  • Insulin / pharmacology
  • Lysosomes / drug effects
  • Lysosomes / metabolism
  • Mechanistic Target of Rapamycin Complex 1 / metabolism*
  • Monomeric GTP-Binding Proteins / metabolism*
  • Neoplasms / metabolism*
  • Neoplasms / pathology*
  • Phosphoric Monoester Hydrolases / metabolism*
  • Protein Binding / drug effects
  • Protein Multimerization / drug effects
  • Resting Phase, Cell Cycle / drug effects
  • Signal Transduction / drug effects
  • Tumor Stem Cell Assay

Substances

  • Amino Acids
  • Insulin
  • Mechanistic Target of Rapamycin Complex 1
  • Phosphoric Monoester Hydrolases
  • RRAGA protein, human
  • NUDT2 protein, human
  • Monomeric GTP-Binding Proteins