Redistribution of regional blood flow after administration of saralasin in salt-depleted dogs

Clin Sci Mol Med Suppl. 1978 Dec:4:243s-246s. doi: 10.1042/cs055243s.

Abstract

1. Salt depletion was produced in five dogs by a low salt diet and daily administration of frusemide for 5 days; a control group of five dogs was placed on the same diet, to which 2.5 g of sodium chloride was added. 2. Saralasin infusion (0.5 microgram min-1 kg-1) reduced mean aortic blood pressure and total peripheral vascular resistance and increased cardiac output in salt-depleted dogs, but did not affect the heart rate and left ventricular dP/dt. 3. Saralasin infusion increased mean aortic blood pressure slightly in normal dogs; other systemic haemodynamic parameters did not change significantly. 4. Saralasin decreased hepatic arterial flow in both normal and salt-depleted dogs, but increased blood flow to left ventricle and kidneys only in salt-depleted dogs. 5. These results suggest that saralasin exerts a partial agonist effect in normal dogs to increase arterial blood pressure, but causes a depressor response during salt depletion because it reverses the vasoconstrictor effect of angiotensin II, particularly on the renal and coronary circulations.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Angiotensin II / analogs & derivatives*
  • Animals
  • Blood Pressure / drug effects
  • Dogs
  • Furosemide / pharmacology
  • Hemodynamics / drug effects*
  • Male
  • Regional Blood Flow / drug effects*
  • Saralasin / pharmacology*
  • Sodium Chloride / metabolism

Substances

  • Angiotensin II
  • Sodium Chloride
  • Furosemide
  • Saralasin