Pathology-targeted cell delivery via injectable micro-scaffold capsule mediated by endogenous TGase

Biomaterials. 2017 May:126:1-9. doi: 10.1016/j.biomaterials.2017.02.021. Epub 2017 Feb 17.

Abstract

Targeted cell delivery to lesion sites via minimally invasive approach remains an unmet need in regenerative medicine to endow satisfactory therapeutic efficacy and minimized side-effects. Here, we rationally designed a pathology-targeted cell delivery strategy leveraging injectable micro-scaffolds as cell-loading capsule and endogenous tissue transglutaminase (TGase) at lesion site as adhesive. Up-regulated TGase post-liver injury catalyzed chemical bonding between the glutamine and lysine residues on liver surface and micro-scaffolds both ex vivo and in vivo, facilitating sufficient adhesion on the pathological liver. Upon intraperitoneal injection, Mesenchymal Stem Cell-loaded capsules, exhibiting cell protection from shear-induced damage and post-transplantation anoikis, adhered to the CCl4-treated liver with a hundred-fold improvement in targeting efficiency (70.72%) compared to free-cell injection, which dramatically improved mice survival (33.3% vs. 0% for free-cell therapy) even with low-dosage treatment. This unique and widely-applicable cell delivery mechanism and strategy hold great promise for transforming cell therapy for refractory diseases.

Keywords: Cell therapy; Endogenous TGase; Micro-scaffold capsule; Pathological liver; Targeted cell delivery.

MeSH terms

  • Animals
  • Biocatalysis
  • Capsules
  • Cell Adhesion
  • Drug Delivery Systems*
  • GTP-Binding Proteins / metabolism*
  • Humans
  • Injections*
  • Liver / injuries
  • Liver / pathology
  • Mesenchymal Stem Cell Transplantation
  • Mesenchymal Stem Cells / cytology
  • Mice, Inbred BALB C
  • Mice, Nude
  • Polyethylene Glycols / chemistry
  • Protein Glutamine gamma Glutamyltransferase 2
  • Tissue Scaffolds / chemistry*
  • Transglutaminases / metabolism*

Substances

  • Capsules
  • Polyethylene Glycols
  • Protein Glutamine gamma Glutamyltransferase 2
  • Transglutaminases
  • GTP-Binding Proteins