Ultrasensitive Measurement of Ca2+ Influx into Lipid Vesicles Induced by Protein Aggregates

Angew Chem Int Ed Engl. 2017 Jun 26;56(27):7750-7754. doi: 10.1002/anie.201700966. Epub 2017 May 5.

Abstract

To quantify and characterize the potentially toxic protein aggregates associated with neurodegenerative diseases, a high-throughput assay based on measuring the extent of aggregate-induced Ca2+ entry into individual lipid vesicles has been developed. This approach was implemented by tethering vesicles containing a Ca2+ sensitive fluorescent dye to a passivated surface and measuring changes in the fluorescence as a result of membrane disruption using total internal reflection microscopy. Picomolar concentrations of Aβ42 oligomers could be observed to induce Ca2+ influx, which could be inhibited by the addition of a naturally occurring chaperone and a nanobody designed to bind to the Aβ peptide. We show that the assay can be used to study aggregates from other proteins, such as α-synuclein, and to probe the effects of complex biofluids, such as cerebrospinal fluid, and thus has wide applicability.

Keywords: Alzheimer's disease; fluorescence imaging; nano-scale biophysics; neurodegeneration; protein aggregation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alzheimer Disease / metabolism
  • Alzheimer Disease / pathology
  • Amyloid beta-Peptides / chemistry
  • Amyloid beta-Peptides / immunology
  • Amyloid beta-Peptides / metabolism
  • Calcium / chemistry
  • Calcium / metabolism*
  • Clusterin / chemistry
  • Clusterin / metabolism
  • Fluorescent Dyes / chemistry
  • Humans
  • Kinetics
  • Lipid Bilayers / chemistry
  • Lipid Bilayers / metabolism*
  • Optical Imaging
  • Protein Aggregates / physiology*
  • Protein Binding
  • Single-Domain Antibodies / immunology

Substances

  • Amyloid beta-Peptides
  • Clusterin
  • Fluorescent Dyes
  • Lipid Bilayers
  • Protein Aggregates
  • Single-Domain Antibodies
  • Calcium