Novel drug and soluble target tolerant antidrug antibody assay for therapeutic antibodies bearing the P329G mutation

Bioanalysis. 2017 Jun;9(11):849-859. doi: 10.4155/bio-2017-0048. Epub 2017 May 18.

Abstract

Aim: Bridging immunoassays for detection of antidrug antibodies (ADAs) are typically susceptible to high concentrations of residual drug. Sensitive drug-tolerant assays are, therefore, needed.

Materials & methods: An immune complex assay to detect ADAs against therapeutic antibodies bearing Pro329Gly mutation was established. The assay uses antibodies specific for the Pro329Gly mutation for capture and human soluble Fcγ receptor for detection.

Results: When compared with a bridging assay, the new assay showed similar precision, high sensitivity to IgG1 ADA and dramatically improved drug tolerance. However, it was not able to detect early (IgM-based) immune responses.

Conclusion: Applied in combination with a bridging assay, the novel assay serves as orthogonal assay for immunogenicity assessment and allows further characterization of ADA responses.

Keywords: ELISA; FcγRI; antidrug antibody; drug tolerance; immune complex assay; immunogenicity; safety assessment; suppressed Fc effector functions; target interference.

MeSH terms

  • Animals
  • Antibodies / analysis*
  • Antibodies / immunology*
  • Antibodies, Monoclonal / administration & dosage
  • Antibodies, Monoclonal / genetics
  • Antibodies, Monoclonal / immunology*
  • Antigen-Antibody Complex / immunology*
  • Drug Tolerance
  • Humans
  • Immunoassay / methods*
  • Immunoglobulin G / administration & dosage
  • Immunoglobulin G / genetics
  • Immunoglobulin G / immunology*
  • Mice
  • Point Mutation
  • Receptors, IgG / immunology*
  • Recombinant Proteins / administration & dosage
  • Recombinant Proteins / genetics
  • Recombinant Proteins / immunology

Substances

  • Antibodies
  • Antibodies, Monoclonal
  • Antigen-Antibody Complex
  • Immunoglobulin G
  • Receptors, IgG
  • Recombinant Proteins