Blockade of interleukin-6 receptor in the periphery promotes rapid and sustained antidepressant actions: a possible role of gut-microbiota-brain axis

Transl Psychiatry. 2017 May 30;7(5):e1138. doi: 10.1038/tp.2017.112.

Abstract

Depression is a common, severe and chronic psychiatric disease. Although the currently available antidepressants have been used in the treatment of depression, their beneficial effects are limited. Accumulating evidence suggests that pro-inflammatory cytokines such as interleukin-6 (IL-6) have an important role in the pathogenesis of depression. This study was undertaken to examine whether anti-mouse IL-6 receptor antibody (MR16-1) induces antidepressant effects in a social defeat stress model. Intravenous injection of MR16-1 induced rapid-onset and long-lasting antidepressant effects in susceptible mice after social defeat stress through its anti-inflammatory actions. In contrast, intracerebroventricular injection of MR16-1 induced no antidepressant effects in susceptible mice. Furthermore, treatment with MR16-1 could significantly normalize alterations in the expression of synaptic proteins (postsynaptic density protein 95 and α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor 1) and dendritic spine density in the brain regions of susceptible mice. Gut microbiota analysis using 16S ribosomal RNA gene sequencing showed that MR16-1 significantly improved decreased Firmicutes/Bacteroidetes ratio in susceptible mice. It also significantly improved decreased levels of Oscillospira in susceptible mice. These findings suggest that peripheral IL-6 has a key role in the pathogenesis of depression and that the blockade of IL-6 receptor in the periphery might have rapid-onset and long-lasting antidepressant effects by normalizing the altered composition of gut microbiota in susceptible mice after social defeat stress. Therefore, the blockade of IL-6 receptor in the periphery shows promise as a novel therapeutic approach for depressed patients with higher IL-6 blood levels.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antidepressive Agents / immunology*
  • Antidepressive Agents / metabolism
  • Cytokines / metabolism
  • Depression / immunology*
  • Depression / metabolism
  • Depressive Disorder / drug therapy
  • Disease Models, Animal
  • Gastrointestinal Microbiome / drug effects*
  • Gastrointestinal Microbiome / genetics
  • Interleukin-6 / antagonists & inhibitors
  • Interleukin-6 / blood*
  • Interleukin-6 / immunology
  • Interleukin-6 / metabolism
  • Interleukin-6 / pharmacology
  • Male
  • Mice
  • Mice, Inbred C57BL / psychology
  • Receptors, Interleukin-6 / antagonists & inhibitors*
  • Stress, Psychological / genetics

Substances

  • Antidepressive Agents
  • Cytokines
  • IL6 protein, human
  • Interleukin-6
  • Receptors, Interleukin-6
  • interleukin-6, mouse