A Polycation Antimicrobial Peptide Mimic without Resistance Buildup against Propionibacterium Acnes

Macromol Biosci. 2017 Sep;17(9). doi: 10.1002/mabi.201700090. Epub 2017 Jun 12.

Abstract

A preliminary study is reported for a polycation antimicrobial peptide (AMP) mimic against Propionibacterium acnes, which is associated with acne vulgaris, a common skin condition. Antibiotics are commonly used against P. acnes but buildup of resistance is well-known. Worse, antibiotic regimens build up resistance for more sensitive bacteria such as Staphylococcus epidermidis. The polycation AMP mimic C12-50, 1, is chosen for the present study as it has been previously shown to have high antimicrobial effectiveness. This study reports that C12-50 is active against P. acnes (strain ATCC 6919) with a minimum inhibitory concentration (MIC) of 6.3 µg mL-1 . To monitor resistance build-up ten passages are conducted with C12-50 against P. acnes. The MIC remains constant with no resistance buildup. Parallel studies with erythromycin confirm previously reported resistance buildup. The results point to a promising pathway to applications for polycation AMP mimics against P. acnes.

Keywords: Propionibacterium acnes; acne; antibiotic resistance; minimum inhibitory concentration.

MeSH terms

  • Acne Vulgaris
  • Anti-Infective Agents / pharmacology
  • Antimicrobial Cationic Peptides / pharmacology*
  • Drug Resistance, Microbial
  • Humans
  • Microbial Sensitivity Tests
  • Polyamines / pharmacology
  • Polyelectrolytes
  • Propionibacterium acnes / drug effects*

Substances

  • Anti-Infective Agents
  • Antimicrobial Cationic Peptides
  • Polyamines
  • Polyelectrolytes
  • polycations