Efficacy of the oral neurokinin-1 receptor antagonist aprepitant for nausea and vomiting induced by cisplatin and carboplatin in Japanese patients with gynecological cancer

J Obstet Gynaecol Res. 2017 Oct;43(10):1613-1620. doi: 10.1111/jog.13415. Epub 2017 Jul 10.

Abstract

Aim: This study was conducted to evaluate the efficacy and the difference in effects of the oral neurokinin-1(NK-1) receptor antagonist aprepitant for chemotherapy-induced nausea/vomiting (CINV) in Japanese patients with gynecological cancer receiving highly emetogenic (cisplatin) and moderately emetogenic (carboplatin) chemotherapy.

Methods: Aprepitant was added during the second course of chemotherapy in Japanese patients with grade ≥ 2 (Common Terminology Criteria for Adverse Events, version 3.0) nausea and vomiting during the first course despite receiving antiemetic therapy (a first-generation 5-hydroxytryptamine 3 receptor antagonist + dexamethasone), and in patients who requested stronger antiemetic therapy despite only having grade 1 nausea and vomiting. The incidence of nausea and vomiting was compared between the first and second courses in each group.

Results: Ninety-six (55.5%) out of 173 patients received add-on therapy with aprepitant. There was a significant increase in the complete response (CR: no vomiting or salvage therapy) rate in the patients receiving aprepitant, with marked improvement being confirmed for delayed CINV. Stratified analysis showed that patients with delayed CINV treated with carboplatin had a significantly higher CR rate, while patients with both acute and delayed CINV treated with cisplatin had significantly higher CR rates. There was a positive correlation between the incidence of nausea and the incidence of vomiting in the patients treated with aprepitant.

Conclusion: The oral NK-1 receptor antagonist aprepitant could be effective for both acute and delayed CINV with cisplatin and for delayed CINV with carboplatin in Japanese gynecological cancer patients.

Keywords: Aprepitant; carboplatin; chemotherapy-induced nausea and vomiting (CINV); cisplatin; gynecological cancer.

MeSH terms

  • Adult
  • Aged
  • Antineoplastic Agents / adverse effects*
  • Aprepitant
  • Carboplatin / adverse effects*
  • Cisplatin / adverse effects*
  • Female
  • Genital Neoplasms, Female / drug therapy*
  • Humans
  • Japan
  • Middle Aged
  • Morpholines / administration & dosage
  • Morpholines / pharmacology*
  • Nausea / chemically induced
  • Nausea / drug therapy*
  • Neurokinin-1 Receptor Antagonists / administration & dosage
  • Neurokinin-1 Receptor Antagonists / pharmacology*
  • Outcome Assessment, Health Care*
  • Vomiting / chemically induced
  • Vomiting / drug therapy*

Substances

  • Antineoplastic Agents
  • Morpholines
  • Neurokinin-1 Receptor Antagonists
  • Aprepitant
  • Carboplatin
  • Cisplatin