How to select a nanosimilar

Ann N Y Acad Sci. 2017 Nov;1407(1):50-62. doi: 10.1111/nyas.13382. Epub 2017 Jul 17.

Abstract

Nanomedicines in the class of nonbiological complex drugs (NBCDs) are becoming increasingly available. Up to 23 nanomedicines have been approved, and approximately 50 are in clinical development. Meanwhile, the first nanosimilars have entered the market through the generic approval pathway, but clinical differences have been observed. Many healthcare professionals may be unaware of this issue and must be informed of these clinically relevant variances. This article provides a tool for rational decision making for the inclusion of nanomedicines into the hospital formulary, including defined criteria for evaluation of substitutability or interchangeability. The tool was generated by conducting a roundtable with an international panel of experts and follows the same thought process that was developed and published earlier for the selection of biologicals/biosimilars. In addition to the existing criteria for biosimilars, a set of seven criteria was identified that specifically apply to nanosimilars. These include (1) particle size and size distribution, (2) particle surface characteristics, (3) fraction of uncaptured bioactive moiety, (4) stability on storage, (5) bioactive moiety uptake and (6) distribution, and (7) stability for ready-to-use preparation. Pharmacists should utilize their pharmaceutical expertise to use the appropriate criteria to evaluate the comparability of the drug to decide on interchangeability or substitutability.

Keywords: hospital formulary; interchange; nanomedicines; nanosimilars; substitution.

MeSH terms

  • Algorithms
  • Biosimilar Pharmaceuticals / pharmacokinetics
  • Biosimilar Pharmaceuticals / standards*
  • Biosimilar Pharmaceuticals / therapeutic use
  • Drug Approval / methods*
  • Drugs, Generic / pharmacokinetics
  • Drugs, Generic / standards*
  • Drugs, Generic / therapeutic use
  • Guidelines as Topic
  • Humans
  • International Cooperation
  • Nanomedicine / methods*
  • Pharmacovigilance
  • Therapeutic Equivalency

Substances

  • Biosimilar Pharmaceuticals
  • Drugs, Generic