Berberine promotes ischemia-induced angiogenesis in mice heart via upregulation of microRNA-29b

Clin Exp Hypertens. 2017;39(7):672-679. doi: 10.1080/10641963.2017.1313853. Epub 2017 Jul 19.

Abstract

Background: Berberine has several preventive effects on cardiovascular diseases. Increased expression of miR-29b has been reported to attenuate cardiac remodeling after myocardial infarction (MI). We hypothesized that berberine via an miR-29b-dependent mechanism promotes angiogenesis and improves heart functions in mice after MI.

Methods: The MI model was established in mice by ligation of left anterior descending coronary artery. The expression of miR-29b was examined by RT-qPCR. Angiogenesis was assessed by immunohistochemistry.

Results: Berberine increased miR-29b expression and promoted cell proliferations and migrations in cultured endothelial cells, which were abolished by miR-29b antagomir or AMP-activated protein kinase inhibitor compound C. In mice following MI, administration of berberine significantly increased miR-29b expressional level, promoted angiogenesis, reduced infarct size, and improved heart functions after 14 postoperative days. Importantly, these in vivo effects of berberine were ablated by antagonism of miR-29b.

Conclusion: Berberine via upregulation of miR-29b promotes ischemia-induced angiogenesis and improves heart functions.

Keywords: AMPK; Akt; angiogenesis; berberine; miR-29b; myocardial infarction.

MeSH terms

  • AMP-Activated Protein Kinases / metabolism
  • Angiogenesis Inducing Agents / pharmacology*
  • Animals
  • Berberine / pharmacology*
  • Cell Proliferation / physiology
  • Heart / drug effects
  • Hypertension / physiopathology
  • Male
  • Mice, Inbred C57BL
  • MicroRNAs / biosynthesis
  • MicroRNAs / drug effects*
  • Myocardial Infarction / physiopathology
  • Transcriptional Activation / physiology
  • Up-Regulation / drug effects
  • Vascular Remodeling / drug effects

Substances

  • Angiogenesis Inducing Agents
  • MicroRNAs
  • Berberine
  • AMP-Activated Protein Kinases