Two new cassane diterpene lactams from the fruits of Caesalpinia mimosoides Lam

Nat Prod Res. 2018 Apr;32(8):875-879. doi: 10.1080/14786419.2017.1365070. Epub 2017 Aug 16.

Abstract

Two new cassane ditepenoid lactams, caesmimotam A (1) and B (2), along with eight known compounds (3-10) were isolated from the fruits of Caesalpinia mimosoides Lam. Their structures were identified by 1D and 2D NMR spectral data. Compounds 1 and 2 were evaluated for their cytotoxicity on HL-60, SMMC-7721, A-549, MCF-7 and SW-480 human cancer cell lines, but they were inactive.

Keywords: Caesalpinia mimosoides; Caesmimotams A and B; Cassane diterpenoid lactam; Leguminaceae.

MeSH terms

  • Antineoplastic Agents, Phytogenic / chemistry
  • Antineoplastic Agents, Phytogenic / pharmacology
  • Caesalpinia / chemistry*
  • Cell Line, Tumor
  • Diterpenes / chemistry*
  • Diterpenes / pharmacology
  • Drug Screening Assays, Antitumor
  • Fruit / chemistry
  • HL-60 Cells
  • Humans
  • Inhibitory Concentration 50
  • Lactams / chemistry*
  • Lactams / pharmacology
  • Magnetic Resonance Spectroscopy
  • Molecular Structure

Substances

  • Antineoplastic Agents, Phytogenic
  • Diterpenes
  • Lactams