New Cassane Diterpenoids from Caesalpinia sappan and their Antiplasmodial Activity

Molecules. 2017 Oct 17;22(10):1751. doi: 10.3390/molecules22101751.

Abstract

One new cassane diterpene possessing an unusual N bridge between C-19 and C-20 named caesalsappanin R (1), as well as another new diterpene caesalsappanin S (2), were isolated from the seeds of Caesalpinia sappanwith methanol extract. Their structures were determined by spectroscopic analysis and examined alongside existing data from prior studies. Their biological activities were profiled by their antiplasmodial activity.

Keywords: Caesalpinia sappan; N bridge; antiplasmodial activity; cassane diterpenes.

MeSH terms

  • Antimalarials / chemistry*
  • Antimalarials / isolation & purification
  • Antimalarials / pharmacology*
  • Caesalpinia / chemistry*
  • Diterpenes / chemistry*
  • Diterpenes / isolation & purification
  • Diterpenes / pharmacology*
  • Inhibitory Concentration 50
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Parasitic Sensitivity Tests
  • Plant Extracts / chemistry
  • Plant Extracts / pharmacology

Substances

  • Antimalarials
  • Diterpenes
  • Plant Extracts