Different structural alterations upregulate in vitro tyrosine kinase activity and transforming potency of the erbB-2 gene

Mol Cell Biol. 1988 Dec;8(12):5570-4. doi: 10.1128/mcb.8.12.5570-5574.1988.

Abstract

Compared with normal erbB-2 gp185, mutant erbB-2 proteins generated by mutations either in the transmembrane domain or by NH2-terminal deletion are able to transform NIH 3T3 cells at a 10- to 100-fold greater efficiency. Mutant proteins of both classes show increased tyrosine kinase activity, suggesting that an abnormal level of receptor-associated tyrosine kinase activity is a major determinant of erbB-2 oncogenic potential.

MeSH terms

  • Animals
  • Cell Transformation, Neoplastic
  • Cells, Cultured
  • Genes*
  • Genes, Regulator*
  • Mice
  • Oncogenes*
  • Protein-Tyrosine Kinases / biosynthesis
  • Protein-Tyrosine Kinases / genetics*
  • Protein-Tyrosine Kinases / metabolism
  • Proto-Oncogene Proteins / biosynthesis
  • Proto-Oncogene Proteins / genetics*
  • Receptor, ErbB-2

Substances

  • Proto-Oncogene Proteins
  • Protein-Tyrosine Kinases
  • Receptor, ErbB-2