A glycerophospholipid-specific pocket in the RVFV class II fusion protein drives target membrane insertion

Science. 2017 Nov 3;358(6363):663-667. doi: 10.1126/science.aal2712.

Abstract

The Rift Valley fever virus (RVFV) is transmitted by infected mosquitoes, causing severe disease in humans and livestock across Africa. We determined the x-ray structure of the RVFV class II fusion protein Gc in its postfusion form and in complex with a glycerophospholipid (GPL) bound in a conserved cavity next to the fusion loop. Site-directed mutagenesis and molecular dynamics simulations further revealed a built-in motif allowing en bloc insertion of the fusion loop into membranes, making few nonpolar side-chain interactions with the aliphatic moiety and multiple polar interactions with lipid head groups upon membrane restructuring. The GPL head-group recognition pocket is conserved in the fusion proteins of other arthropod-borne viruses, such as Zika and chikungunya viruses, which have recently caused major epidemics worldwide.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cell Membrane / virology*
  • Chikungunya virus / chemistry
  • Chikungunya virus / ultrastructure
  • Cholesterol / chemistry
  • Conserved Sequence
  • Crystallography, X-Ray
  • Glycerophospholipids / chemistry*
  • Humans
  • Livestock / virology
  • Molecular Dynamics Simulation
  • Mutagenesis, Site-Directed
  • Protein Conformation
  • Rift Valley fever virus / chemistry*
  • Rift Valley fever virus / genetics
  • Rift Valley fever virus / ultrastructure
  • Viral Fusion Proteins / chemistry*
  • Viral Fusion Proteins / genetics
  • Viral Fusion Proteins / ultrastructure
  • Zika Virus / chemistry
  • Zika Virus / ultrastructure

Substances

  • Glycerophospholipids
  • Viral Fusion Proteins
  • Cholesterol