Pulsed electric field-assisted sensitization of multidrug-resistant Candida albicans to antifungal drugs

Future Microbiol. 2018 Apr:13:535-546. doi: 10.2217/fmb-2017-0245. Epub 2017 Dec 11.

Abstract

Aim: Determine the influence of pH on the inactivation efficiency of Candida albicans in pulsed electric fields (PEF) and evaluate the possibilities for sensitization of a drug-resistant strain to antifungal drugs.

Materials & methods: The effects of PEF (2.5-25 kVcm-1) with fluconazole, terbinafine and naftifine were analyzed at a pH range of 3.0-9.0. Membrane permeabilization was determined by flow cytometry and propidium iodide.

Results: PEF induced higher inactivation of C. albicans at low pH and increased sensitivity to terbinafine and naftifine to which the strain was initially resistant. Up to 5 log reduction in cell survival was achieved.

Conclusion: A proof of concept that electroporation can be used to sensitize drug-resistant microorganisms was presented, which is promising for treating biofilm-associated infections.

Keywords: biofilms; electroporation; inactivation; yeast.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Allylamine / analogs & derivatives
  • Allylamine / chemistry
  • Allylamine / pharmacokinetics
  • Antifungal Agents / chemistry
  • Antifungal Agents / pharmacokinetics*
  • Biofilms / drug effects
  • Candida albicans / drug effects*
  • Candida albicans / physiology
  • Cell Membrane Permeability / drug effects*
  • Drug Resistance, Multiple, Fungal*
  • Electric Stimulation
  • Electrochemical Techniques*
  • Fluconazole / chemistry
  • Fluconazole / pharmacokinetics
  • Humans
  • Hydrogen-Ion Concentration
  • Naphthalenes / chemistry
  • Naphthalenes / pharmacokinetics
  • Propidium / chemistry
  • Terbinafine

Substances

  • Antifungal Agents
  • Naphthalenes
  • Propidium
  • Allylamine
  • naftifine
  • Fluconazole
  • Terbinafine