Quercetin protects against chronic prostatitis in rat model through NF-κB and MAPK signaling pathways

Prostate. 2018 Aug;78(11):790-800. doi: 10.1002/pros.23536. Epub 2018 Apr 13.

Abstract

Background: Chronic Prostatitis/Chronic Pelvic Pain Syndrome (CP/CPPS) is a common disease of urology, of which the pathogenesis and therapy remain to be further elucidated. Quercetin has been reported to improve the symptoms of CP/CPPS patients. We aimed to verify the therapeutic effect of quercetin on CP/CPPS and identify the mechanism responsible for it.

Methods: A novel CP/CPPS model induced with Complete Freund Adjuvant in Sprague Dawley rats was established and the prostates and blood specimens were harvested for further measurement after oral administration of quercetin for 4 weeks.

Results: Increased prostate index and infiltration of lymphocytes, up-regulated expression of IL-1β, IL-2, IL-6, IL-17A, MCP1, and TNFα, decreased T-SOD, CAT, GSH-PX, and increased MDA, enhanced phosphorylation of NF-κB, P38, ERK1/2, and SAPK/JNK were detected in CP/CPPS rat model. Quercetin was identified to ameliorate the histo-pathologic changes, decrease the expression of pro-inflammatory cytokines IL-1β, IL-2, IL-6, IL-17A, MCP1, and TNFα, improve anti-oxidant capacity, and suppress the phosphorylation of NF-κB and MAPKs.

Conclusions: Quercetin has specific protective effect on CP/CPPS, which is mediated by anti-inflammation, anti-oxidation, and at least partly through NF-κB and MAPK signaling pathways.

Keywords: Chronic Prostatitis/Chronic Pelvic Pain Syndrome; anti-inflammation; anti-oxidation; quercetin; signal pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / metabolism
  • Antioxidants / pharmacology
  • Chemokine CCL2 / metabolism
  • Chronic Disease / drug therapy
  • Chronic Disease / prevention & control
  • Disease Models, Animal
  • Interleukins / metabolism
  • Lipid Peroxidation / drug effects
  • MAP Kinase Signaling System / drug effects*
  • Male
  • NF-kappa B / metabolism*
  • Prostate / drug effects
  • Prostate / metabolism
  • Prostate / pathology
  • Prostatitis / drug therapy
  • Prostatitis / metabolism
  • Prostatitis / pathology
  • Prostatitis / prevention & control*
  • Quercetin / pharmacology*
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Antioxidants
  • Chemokine CCL2
  • Interleukins
  • NF-kappa B
  • Tumor Necrosis Factor-alpha
  • Quercetin