Non-canonical functions of the RB protein in cancer

Nat Rev Cancer. 2018 Jul;18(7):442-451. doi: 10.1038/s41568-018-0008-5.

Abstract

The canonical model of RB-mediated tumour suppression developed over the past 30 years is based on the regulation of E2F transcription factors to restrict cell cycle progression. Several additional functions have been proposed for RB, on the basis of which a non-canonical RB pathway can be described. Mechanistically, the non-canonical RB pathway promotes histone modification and regulates chromosome structure in a manner distinct from cell cycle regulation. These functions have implications for chemotherapy response and resistance to targeted anticancer agents. This Opinion offers a framework to guide future studies of RB in basic and clinical research.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Antineoplastic Agents / therapeutic use
  • Cell Proliferation
  • Chromatin / metabolism
  • Chromosome Structures*
  • DNA Repair / physiology
  • Drug Resistance, Neoplasm*
  • E2F Transcription Factors / metabolism
  • Epigenesis, Genetic
  • Genomic Instability
  • Histone Code*
  • Humans
  • Molecular Targeted Therapy
  • Neoplasms / drug therapy
  • Neoplasms / genetics
  • Neoplasms / metabolism*
  • Phosphorylation
  • Retinoblastoma Protein / metabolism*

Substances

  • Antineoplastic Agents
  • Chromatin
  • E2F Transcription Factors
  • Retinoblastoma Protein