Impact of Obesity on Fosphenytoin Volume of Distribution in Pediatric Patients

J Child Neurol. 2018 Jul;33(8):534-536. doi: 10.1177/0883073818770801. Epub 2018 May 1.

Abstract

The impact of body habitus on fosphenytoin pharmacokinetics is poorly understood in pediatric patients. This retrospective, single-center review examined differences in fosphenytoin volume of distribution (VD) between children with normal and obese body habitus. From 2013 to 2015, patients 2 to 18 years of age who received a loading dose of fosphenytoin were identified. Thirty-seven patients met inclusion criteria. Mean total serum phenytoin concentration was 25.3 ± 6.5 μg/mL in the nonobese group and 29.5 ± 7.6 μg/mL in the obese group ( P = .09). VD was not significantly different between obese and nonobese groups, 0.92 ± 0.26 L/kg and 0.97 ± 0.48 L/kg ( P = .76), respectively. In contrast to adult studies, these data suggest that fosphenytoin dose adjustments for obese children may be unnecessary.

Keywords: antiepileptic drugs; children; pediatric; status epilepticus; treatment.

MeSH terms

  • Adolescent
  • Anticonvulsants / blood*
  • Anticonvulsants / therapeutic use
  • Child
  • Child, Preschool
  • Female
  • Humans
  • Male
  • Obesity / blood*
  • Obesity / complications
  • Phenytoin / analogs & derivatives*
  • Phenytoin / blood
  • Phenytoin / therapeutic use
  • Retrospective Studies
  • Status Epilepticus / blood
  • Status Epilepticus / complications
  • Status Epilepticus / drug therapy

Substances

  • Anticonvulsants
  • Phenytoin
  • fosphenytoin