A new 5'-nucleotidase inhibitor, nucleoticidin. I. Taxonomy, fermentation, isolation and biological properties

J Antibiot (Tokyo). 1985 Feb;38(2):153-6. doi: 10.7164/antibiotics.38.153.

Abstract

A new 5'-nucleotidase inhibitor named nucleoticidin was produced by Pseudomonas sp. YM-3229G. It was isolated from a fermentation broth by trichloroacetic acid extraction, ethanol precipitation and Dowex 1 and DEAE-52 column chromatography. It inhibited 5'-nucleotidase activity of snake venom and rat liver membrane. It also showed antitumor activity against solid type Sarcoma 180.

MeSH terms

  • Animals
  • Anti-Bacterial Agents / isolation & purification*
  • Anti-Bacterial Agents / pharmacology
  • Antibiotics, Antineoplastic / isolation & purification
  • Antibiotics, Antineoplastic / pharmacology
  • Cell Survival / drug effects
  • Fermentation
  • Liver / enzymology
  • Nucleotidases / antagonists & inhibitors*
  • Pseudomonas / metabolism
  • Rats
  • Sarcoma, Experimental / metabolism
  • Snake Venoms / antagonists & inhibitors
  • Soil Microbiology

Substances

  • Anti-Bacterial Agents
  • Antibiotics, Antineoplastic
  • Snake Venoms
  • Nucleotidases
  • nucleotidase