Nanoemulsion-Loaded Hydrogels for Topical Administration of Pentyl Gallate

AAPS PharmSciTech. 2018 Aug;19(6):2672-2678. doi: 10.1208/s12249-018-1099-8. Epub 2018 Jun 25.

Abstract

The aim of this study is to describe the development of nanoemulsion-loaded hydrogels to deliver pentyl gallate (PG), a gallic acid n-alkyl ester, through the skin. PG is an antioxidant agent; however, it seems to be a promising agent for herpis labialis treatment. Aristoflex AVC® and chitosan were used as gelling agents for nanoemulsion thickening. The developed formulations presented suitable PG content (94.4-100.3% w/w), nanometric droplet sizes (162-297 nm), high zeta potentials, and a non-Newtonian pseudoplastic behavior. Both vehicles neither enhanced PG penetration nor delayed its release from the nanoemulsion. Formulations remained physically stable at 8°C during 3 months of storage.

Keywords: hydrogel; nanoemulsion; pentyl gallate.

MeSH terms

  • Administration, Topical
  • Animals
  • Antioxidants / administration & dosage
  • Antioxidants / metabolism
  • Drug Compounding
  • Emulsions / administration & dosage*
  • Emulsions / metabolism
  • Gallic Acid / administration & dosage
  • Gallic Acid / analogs & derivatives*
  • Gallic Acid / metabolism
  • Hydrogels / administration & dosage*
  • Hydrogels / metabolism
  • Nanoparticles / administration & dosage*
  • Nanoparticles / metabolism
  • Organ Culture Techniques
  • Skin / drug effects
  • Skin / metabolism
  • Skin Absorption / drug effects*
  • Skin Absorption / physiology
  • Swine

Substances

  • Antioxidants
  • Emulsions
  • Hydrogels
  • pentyl gallate
  • Gallic Acid