[Medical treatment of small cell lung cancer: Can we leave the area of cisplatin-etoposide?]

Bull Cancer. 2018 Oct;105(10):955-966. doi: 10.1016/j.bulcan.2018.05.014. Epub 2018 Aug 9.
[Article in French]

Abstract

Small cell lung cancer accounts for 14% of all lung cancers. It remains a major challenge for oncology as the progresses made in the past three decades are modest. After a rapid overview of current knowledge regarding somatic genomic alterations, this state-of-art addresses pathways to improve small-cell lung cancer outcome such as the targeting of DNA damage repair mechanisms firstly anti-PARPs, inhibitory molecules of EZH2, derepression of the NOTCH pathway, rovalbituzumab-tesirine, inhibition of serine/threonine Aurora A kinase, temozolomide and its dependence on methylation of the MGMT promoter. This first chapter suggests the beginning of precision medicine in small cell lung cancer. The last section focuses on the development of immuno-oncological agents and the information collected from phase 1 and 2 studies: the low intensity of PD-L1 tissue expression and the possible relationship of the activity of these agents as a function of tumor mutational burden are pointed out.

Keywords: Alisertib; Anti-PARP; Atezolizumab; Atézolizumab; Aurora A; C-myc; Cancer du poumon à petites cellules; EZH2; Extensive-disease; Maladie étendue; NOTCH; Nivolumab; P53; Pembrolizumab; RB1; Rovalpituzumab–teserine; Rovalpituzumab–tésirine; SLNF-11; Small cell lung cancer; Veliparib; Véliparib.

Publication types

  • Review

MeSH terms

  • Antibodies, Monoclonal, Humanized / therapeutic use
  • Antineoplastic Agents / therapeutic use*
  • Aurora Kinase A / antagonists & inhibitors
  • Benzodiazepinones / therapeutic use
  • DNA Damage
  • DNA Modification Methylases / metabolism
  • DNA Repair
  • DNA Repair Enzymes / metabolism
  • Dacarbazine / analogs & derivatives
  • Dacarbazine / therapeutic use
  • Enhancer of Zeste Homolog 2 Protein / antagonists & inhibitors
  • Humans
  • Immunoconjugates / therapeutic use
  • Lung Neoplasms / drug therapy*
  • Lung Neoplasms / genetics
  • Lung Neoplasms / pathology
  • Poly(ADP-ribose) Polymerase Inhibitors / therapeutic use
  • Protein Serine-Threonine Kinases / antagonists & inhibitors
  • Receptors, Notch / metabolism
  • Small Cell Lung Carcinoma / drug therapy*
  • Small Cell Lung Carcinoma / genetics
  • Small Cell Lung Carcinoma / pathology
  • Temozolomide
  • Tumor Suppressor Proteins / metabolism

Substances

  • Antibodies, Monoclonal, Humanized
  • Antineoplastic Agents
  • Benzodiazepinones
  • Immunoconjugates
  • Poly(ADP-ribose) Polymerase Inhibitors
  • Receptors, Notch
  • Tumor Suppressor Proteins
  • rovalpituzumab tesirine
  • Dacarbazine
  • DNA Modification Methylases
  • EZH2 protein, human
  • Enhancer of Zeste Homolog 2 Protein
  • MGMT protein, human
  • Aurora Kinase A
  • Protein Serine-Threonine Kinases
  • DNA Repair Enzymes
  • Temozolomide