Resistance of high fitness hepatitis C virus to lethal mutagenesis

Virology. 2018 Oct:523:100-109. doi: 10.1016/j.virol.2018.07.030. Epub 2018 Aug 11.

Abstract

Viral fitness quantifies the degree of virus adaptation to a given environment. How viral fitness can influence the mutant spectrum complexity of a viral quasispecies subjected to lethal mutagenesis has not been investigated. Here we document that two high fitness hepatitis C virus populations display higher resistance to the mutagenic nucleoside analogues favipiravir and ribavirin than their parental, low fitness HCV. All populations, however, exhibited a mutation transition bias indicative of active mutagenesis. Resistance to the analogues was associated with a limited expansion of mutant spectrum complexity, as evidenced by several diversity indices used to characterize mutant spectra. The results are consistent with a replicative site-drug competition mechanism that was previously proposed for HCV fitness-associated resistance to non-mutagenic inhibitors. Other alternative, non-mutually exclusive mechanisms are considered. The results introduce viral fitness as a relevant parameter to evaluate the response of viruses to lethal mutagenesis, with implications for antiviral designs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amides / pharmacology*
  • Antiviral Agents / pharmacology*
  • Cell Line, Tumor
  • Drug Resistance, Viral / genetics*
  • Genetic Fitness / drug effects
  • Hepacivirus / drug effects*
  • Hepacivirus / genetics
  • Hepacivirus / growth & development
  • Hepatocytes / drug effects
  • Hepatocytes / virology
  • Humans
  • Mutagenesis*
  • Mutation
  • Pyrazines / pharmacology*
  • Ribavirin / pharmacology*
  • Serial Passage

Substances

  • Amides
  • Antiviral Agents
  • Pyrazines
  • Ribavirin
  • favipiravir