Depression of spike adaptation and afterhyperpolarization by 4-aminopyridine in hippocampal neurons

Neurosci Lett. 1986 Apr 24;65(3):316-20. doi: 10.1016/0304-3940(86)90281-8.

Abstract

In guinea pig hippocampal slices, 4-aminopyridine (4-AP) in concentrations of 100-500 microM reduced the adaptation of CA3 pyramidal neurons to depolarizing stimuli, resulting in a prolongation of repetitive firing during injection of long-lasting depolarizing currents. Concurrently, there was a decrease in the 'sag' of potential after spike bursts. Furthermore, 4-AP decreased or abolished the hyperpolarizing potential (the afterhyperpolarization) which normally followed repetitive firing of the neurons. The findings suggest that 4-AP could interfere with the Ca2+-activated K+ current in hippocampal CA3 pyramidal neurons.

MeSH terms

  • 4-Aminopyridine
  • Action Potentials* / drug effects
  • Adaptation, Physiological / drug effects
  • Aminopyridines / pharmacology*
  • Animals
  • Electric Stimulation
  • Guinea Pigs
  • Hippocampus / drug effects
  • Hippocampus / physiology*
  • Membrane Potentials / drug effects
  • Neural Inhibition / drug effects*

Substances

  • Aminopyridines
  • 4-Aminopyridine