Randomized trial of vonoprazan-based versus proton-pump inhibitor-based third-line triple therapy with sitafloxacin for Helicobacter pylori

J Gastroenterol Hepatol. 2019 Apr;34(4):686-692. doi: 10.1111/jgh.14456. Epub 2018 Sep 21.

Abstract

Background and aim: This was a prospective, randomized trial of the efficacy of vonoprazan-based and proton-pump inhibitor-based 7-day triple regimens with amoxicillin and sitafloxacin as a third-line therapy for eradicating Helicobacter pylori after failure of clarithromycin-based and metronidazole-based first-line and second-line therapy.

Methods: We enrolled 63 patients positive for H. pylori in whom first-line and second-line regimens for eradicating failed. Patients were randomized to the V-AS group (vonoprazan 20-mg bid, amoxicillin 750-mg bid, and sitafloxacin 100-mg bid for 7 days) or PPI-AS group (esomeprazole 20-mg bid, rabeprazole 10-mg bid, or lansoprazole 30-mg bid; amoxicillin 750-mg bid; and sitafloxacin 100-mg bid for 7 days). We assessed the outcome of eradication therapy using the 13 C-urea breath test. We evaluated safety using patient questionnaires. This study was registered in the UMIN Clinical Trials Registry (UMIN000016336).

Results: The intention-to-treat and per-protocol eradication rates of V-AS were 75.8% (95% confidence interval [CI]: 57.7-88.9%) and 83.3% (95% CI: 65.3-94.4%), respectively. The respective eradication rates of PPI-AS were 53.3% (95% CI: 34.3-71.7%) and 57.1% (95% CI: 37.2-75.5%). In per-protocol analyses, the eradication rate of the V-AS group was significantly higher than that of the PPI-AS group (P = 0.043); however, no significant differences were observed in intention-to-treat analyses (P = 0.071). Questionnaire scores did not differ significantly between the groups.

Conclusions: The findings suggest that 7-day triple therapy with vonoprazan, amoxicillin, and sitafloxacin is more effective than proton-pump inhibitor, amoxicillin, and sitafloxacin as a third-line regimen for eradicating H. pylori.

Keywords: 7-day triple therapy; Helicobacter pylori; amoxicillin; sitafloxacin; vonoprazan.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • Amoxicillin / administration & dosage*
  • Anti-Bacterial Agents / administration & dosage*
  • Clarithromycin / administration & dosage
  • Drug Therapy, Combination
  • Esomeprazole / administration & dosage
  • Female
  • Fluoroquinolones / administration & dosage*
  • Gastritis / drug therapy*
  • Gastritis / microbiology*
  • Humans
  • Lansoprazole / administration & dosage
  • Male
  • Metronidazole / administration & dosage
  • Middle Aged
  • Prospective Studies
  • Proton Pump Inhibitors / administration & dosage*
  • Pyrroles / administration & dosage*
  • Rabeprazole / administration & dosage
  • Sulfonamides / administration & dosage*
  • Treatment Failure
  • Treatment Outcome

Substances

  • 1-(5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl)-N-methylmethanamine
  • Anti-Bacterial Agents
  • Fluoroquinolones
  • Proton Pump Inhibitors
  • Pyrroles
  • Sulfonamides
  • Lansoprazole
  • Metronidazole
  • Rabeprazole
  • Amoxicillin
  • sitafloxacin
  • Clarithromycin
  • Esomeprazole