Curcumin analogs: Their roles in pancreatic cancer growth and metastasis

Int J Cancer. 2019 Jul 1;145(1):10-19. doi: 10.1002/ijc.31867. Epub 2018 Dec 11.

Abstract

Curcumin is a polyphenolic constituent of turmeric that is known to have various molecular effects in preclinical models, leading to prevention and anticancer properties. In clinical trials, curcumin has failed to demonstrate activity against pancreatic cancer possibly due to its low bioavailability and potency. Using the curcumin molecular model, our group and others have synthesized several analogs with better bioavailability and higher potency in pancreatic cancer in vitro and xenograft models. This mini review summarizes some of the known molecular effects of curcumin analogs and their potential role as novel therapeutics for pancreatic cancer.

Keywords: analogs; curcumin; growth; metastasis; pancreatic cancer.

Publication types

  • Review

MeSH terms

  • Animals
  • Curcumin / analogs & derivatives*
  • Curcumin / pharmacokinetics
  • Curcumin / pharmacology*
  • Curcumin / therapeutic use
  • Humans
  • Pancreatic Neoplasms / drug therapy*
  • Pancreatic Neoplasms / metabolism

Substances

  • Curcumin