A Natural Phenolic Compound Quercetin Showed the Usefulness by Targeting Inflammatory, Oxidative Stress Markers and Augment 5-HT Levels in One of the Animal Models of Depression in Mice

Drug Res (Stuttg). 2019 Jul;69(7):392-400. doi: 10.1055/a-0748-5518. Epub 2018 Oct 8.

Abstract

Aim: In the present study quercetin was studied for its role in inflammation, oxidative stress markers and 5-HT levels in unpredictable chronic mild stress (UCMS) animal model of depression.

Materials and methods: The mice were randomized into different groups trained for UCMS protocol followed by different drug treatments. Treatments were started after 2 weeks from the start of UCMS protocol and continued up to 6 weeks. The behavioral tests such as modified forced swimming (MFST), tail suspension (TST) and open field tests were performed on week 6, at least 24 h after the last drug treatment. Behavioral tests were preceded following animal sacrifice for biochemical estimations.

Results: A significant decrease in swimming, climbing times and increase in immobility time in MFST and TST was observed in UCMS group. Administration of quercetin (25 mg/kg per orally (p.o) reversed these times in MFST and TST. A decrease in no. of field crossing, time spent in centre and no. of rearing were observed in UCMS group. Quercetin reduced these observations in open field test. There was a decrease in superoxide dismutase (SOD), glutathione (GSH), catalase and 5 HT levels in the brain tissue. Quercetin treatment significantly augmented SOD, GSH, catalase and 5 HT levels. Glutamate, TNF-α and IL-6 levels were increased in UCMS group while quercetin decreased these cytokines.

Conclusion: Quercetin resulted antidepressant-like effect by its antioxidant, anti-inflammatory activities, reduced excitotoxicity and augmented 5 HT levels. This pointed out the usefulness of this phenolic compound as adjuvent drug along with other antidepressant drugs.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology
  • Anti-Inflammatory Agents / therapeutic use
  • Antidepressive Agents / pharmacology*
  • Antidepressive Agents / therapeutic use
  • Antioxidants / pharmacology
  • Antioxidants / therapeutic use
  • Behavior, Animal / drug effects
  • Biomarkers / analysis
  • Biomarkers / metabolism
  • Brain / drug effects*
  • Brain / immunology
  • Brain / pathology
  • Depression / drug therapy*
  • Depression / etiology
  • Depression / pathology
  • Disease Models, Animal
  • Humans
  • Inflammation / drug therapy*
  • Inflammation / pathology
  • Male
  • Mice
  • Oxidative Stress / drug effects
  • Quercetin / pharmacology*
  • Quercetin / therapeutic use
  • Serotonin / analysis
  • Serotonin / metabolism
  • Stress, Psychological / complications
  • Treatment Outcome

Substances

  • Anti-Inflammatory Agents
  • Antidepressive Agents
  • Antioxidants
  • Biomarkers
  • Serotonin
  • Quercetin