The core structure characterization and of ginseng neutral polysaccharide with the immune-enhancing activity

Int J Biol Macromol. 2019 Feb 15:123:713-722. doi: 10.1016/j.ijbiomac.2018.11.140. Epub 2018 Nov 17.

Abstract

The study aims to clarify the structural domain required for the immune enhancement of ginseng neutral polysaccharide (GPN). GPN was first obtained through water extraction and ion-exchange chromatography from Panax ginseng. GPN was hydrolyzed by α-amylase for 24 h and fractionated through gel permeation chromatography to give two final fragments GPNE-I and GPNE-II, with molecular weight of 8.03 × 104 Da for GPNE-I and 3.15 × 104 Da for respectively. FT-IR, methylation and 1D/2D NMR analysis demonstrated that GPNE-I was a heteropolysaccharide consisting mainly of a glucan domain and type I and II arabinogalactans (AG-I and AG-II). GPNE II was a glucan consisting of (1 → 4)-α-d-Glcp backbone with a substitution at O-6 on every two residues. (1 → 3)-α-d-Glcp and (1 → 6)-α-d-Glcp were located at the branches. In the two fractions, both α- and β-t-Glcp as reductive terminals and →4)-α-Glcp as a non-reducing end were detected. The branching degrees of GPNE-I and GPNE-II were 38.17% and 50.78%, respectively. Immunological experiments revealed that GPNE-I exhibited more effectively stimulated lymphocyte proliferation than GPN and GPNE-II, indicating the former showed potential for immunomodulators applications, indicating that GPNE-I might be the core active domain and necessary for GPN to promote lymphocyte proliferation.

Keywords: Immunostimulating activity; Neutral polysaccharides; Panax ginseng; Structure.

MeSH terms

  • Cell Proliferation / drug effects
  • Glucans / chemistry*
  • Glucans / pharmacology
  • Immunologic Factors / chemistry*
  • Immunologic Factors / immunology
  • Immunologic Factors / isolation & purification
  • Lymphocytes / drug effects
  • Magnetic Resonance Spectroscopy
  • Panax / chemistry*
  • Plant Extracts / chemistry
  • Plant Extracts / pharmacology
  • Polysaccharides / chemistry*
  • Polysaccharides / isolation & purification
  • Polysaccharides / pharmacology
  • Spectroscopy, Fourier Transform Infrared
  • Water / chemistry

Substances

  • Glucans
  • Immunologic Factors
  • Plant Extracts
  • Polysaccharides
  • Water