Using Nrf2/antioxidant response element-dependent signaling to assess the toxicity potential of fly ash particles

Ecotoxicol Environ Saf. 2019 Apr 15:170:172-179. doi: 10.1016/j.ecoenv.2018.11.093. Epub 2018 Dec 5.

Abstract

Epidemiological studies have demonstrated an association between ambient particulate pollution and adverse health effects in humans. The antioxidant-responsive element (ARE) cytoprotective system mediated by the transcription factor NF-E2 p45-related factor 2 (Nrf2) serves as a primary defense against the oxidative stress triggered by particulate matter. In this study, using a cell-based ARE-reporter assay, the fine fractions of the fly ash collected from the municipal solid waste incinerators at four cities in China were examined for their ability to activate Nrf2/ARE signaling. We found that, at a non-lethal dose, all the fly ash samples were able to activate the ARE-reporter gene in a dose- and redox-dependent manner, and this was correlated with their cytotoxicity and their ability to induce DNA damage. Study of the kinetics revealed that fly ash particles elicited a prolonged activation of the ARE-reporter activity. Upon exposure to the particles, the ARE-luciferase activity significantly increased in 2 h, reached a peak at 24 h, and remained high level at 72 h. This was in contrast to the transient activation of the ARE-reporter gene triggered by the Nrf2 activators tert-butylhydroquinone and sulforaphane, while ARE-luciferase activity dropped to the basal level at 72 h from the peak at 24 h. These results demonstrate the robustness of using cell-based ARE-reporter assays to evaluate the oxidative potential of fly ash. Our novel findings suggest that the sustained activation of the Nrf2/ARE signaling pathway induced by fly ash particles perturbs cellular redox homeostasis, which in turn contributes to toxicity.

Keywords: Cell based assay; Fly ash particle; Nrf2/ARE; Oxidative stress.

MeSH terms

  • Antioxidant Response Elements / drug effects*
  • Cell Survival / drug effects
  • China
  • Coal Ash / toxicity*
  • DNA Damage / drug effects
  • Dose-Response Relationship, Drug
  • Humans
  • Hydroquinones
  • Incineration
  • Isothiocyanates
  • MCF-7 Cells
  • NF-E2-Related Factor 2 / genetics
  • NF-E2-Related Factor 2 / metabolism*
  • Oxidation-Reduction / drug effects
  • Oxidative Stress / drug effects
  • Particulate Matter / toxicity
  • Signal Transduction*
  • Sulfoxides

Substances

  • Coal Ash
  • Hydroquinones
  • Isothiocyanates
  • NF-E2-Related Factor 2
  • NFE2L2 protein, human
  • Particulate Matter
  • Sulfoxides
  • 2-tert-butylhydroquinone
  • sulforaphane