Camellia japonica oil suppressed asthma occurrence via GATA-3 & IL-4 pathway and its effective and major component is oleic acid

Phytomedicine. 2019 Apr:57:84-94. doi: 10.1016/j.phymed.2018.12.004. Epub 2018 Dec 10.

Abstract

Background: In December 2016, WHO released a report stating that in 2015 there were 383,000 deaths caused by asthma and 235 million people suffering from asthma. As there are many adverse effects associated with the currently-used asthma drugs, new anti-asthmatic drugs need to be developed.

Purpose: In order to find new drug candidates with safe and low side effects, the anti-asthmatic function and mechanism of C. japonica oil were evaluated, and its active ingredients were analyzed for use in an ovalbumin asthma murine model.

Study design and methods: The study consisted of six groups: control; ovalbumin group; and dexamethasone group as a positive control; and 10, 100, and 500 mg/kg C. japonica oil treatment groups. In order to measure the anti-asthmatic effect of C. japonica oil, WBC and differential cell count in BALF, IgE in serum, morphological changes in pulmonary system, and gene and protein levels such as IFN-γ, IL-12p40, IL-4, IL-5, IL-6, TNF-α, and IL-6 were all evaluated.

Results: C. japonica oil had an anti-asthmatic effect and significantly controlled eosinophil in BALF, Th2-related factors such as GATA-3 that is Th2 cell transcription factor, IL-4, IL-5, and IL-13, and TNF-α in the lung. It also dose-dependently modulated inflammatory cells, T-bet, IL-12p40, and IL-6. Oleci acid was the major gradient (52.89%) in C. japonica oil and also had anti-asthmatic effects such as the downregulation of inflammatory cells, WBC, and eosinophil in BALF, IgE in serum, and morphological changes in the lung.

Conclusion: We concluded that C. japonica oil is a new anti-asthmatic drug candidate and that oleic acid is the major anti-asthmatic ingredient in C. japonica oil.

Keywords: C. japonica oil; Oleic acid; Ovalbumin-induced asthma model; Th2-related factors.

MeSH terms

  • Animals
  • Anti-Asthmatic Agents / chemistry
  • Anti-Asthmatic Agents / pharmacology*
  • Asthma / drug therapy*
  • Asthma / metabolism
  • Bronchoalveolar Lavage Fluid
  • Camellia / chemistry*
  • Cytokines / metabolism
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Eosinophils / drug effects
  • Female
  • GATA3 Transcription Factor / metabolism
  • Interleukin-4 / metabolism
  • Lung / drug effects
  • Lung / metabolism
  • Mice, Inbred BALB C
  • Oleic Acid / analysis
  • Plant Oils / administration & dosage
  • Plant Oils / chemistry
  • Plant Oils / pharmacology*

Substances

  • Anti-Asthmatic Agents
  • Cytokines
  • GATA3 Transcription Factor
  • Gata3 protein, mouse
  • Plant Oils
  • Interleukin-4
  • Oleic Acid