Structural Snapshots of 26S Proteasome Reveal Tetraubiquitin-Induced Conformations

Mol Cell. 2019 Mar 21;73(6):1150-1161.e6. doi: 10.1016/j.molcel.2019.01.018. Epub 2019 Feb 18.

Abstract

The 26S proteasome is the ATP-dependent protease responsible for regulating the proteome of eukaryotic cells through degradation of mainly ubiquitin-tagged substrates. In order to understand how proteasome responds to ubiquitin signal, we resolved an ensemble of cryo-EM structures of proteasome in the presence of K48-Ub4, with three of them resolved at near-atomic resolution. We identified a conformation with stabilized ubiquitin receptors and a previously unreported orientation of the lid, assigned as a Ub-accepted state C1-b. We determined another structure C3-b with localized K48-Ub4 to the toroid region of Rpn1, assigned as a substrate-processing state. Our structures indicate that tetraUb induced conformational changes in proteasome could initiate substrate degradation. We also propose a CP gate-opening mechanism involving the propagation of the motion of the lid to the gate through the Rpn6-α2 interaction. Our results enabled us to put forward a model of a functional cycle for proteasomes induced by tetraUb and nucleotide.

Keywords: K48-Ub(4); Ub-bound; cryo-EM; proteasome.

Publication types

  • Research Support, Non-U.S. Gov't
  • Video-Audio Media

MeSH terms

  • Allosteric Regulation
  • Animals
  • Binding Sites
  • Cryoelectron Microscopy
  • DNA-Binding Proteins / genetics
  • DNA-Binding Proteins / metabolism
  • Endopeptidases / genetics
  • Endopeptidases / metabolism
  • Humans
  • Models, Molecular
  • Proteasome Endopeptidase Complex / genetics
  • Proteasome Endopeptidase Complex / metabolism*
  • Proteasome Endopeptidase Complex / ultrastructure
  • Protein Binding
  • Protein Conformation
  • Proteolysis
  • Saccharomyces cerevisiae / enzymology*
  • Saccharomyces cerevisiae / genetics
  • Saccharomyces cerevisiae / ultrastructure
  • Saccharomyces cerevisiae Proteins / genetics
  • Saccharomyces cerevisiae Proteins / metabolism*
  • Saccharomyces cerevisiae Proteins / ultrastructure
  • Structure-Activity Relationship
  • Ubiquitin / metabolism*
  • Ubiquitin / ultrastructure
  • Ubiquitination

Substances

  • DNA-Binding Proteins
  • RAD23 protein, S cerevisiae
  • Saccharomyces cerevisiae Proteins
  • Ubiquitin
  • Endopeptidases
  • Rpn6 protein, S cerevisiae
  • Proteasome Endopeptidase Complex
  • ATP dependent 26S protease
  • UBP6 protein, S cerevisiae