The asymmetric construction of CF3-containing spiro-thiazolone-pyrrolidine compounds via [3 + 2] cycloaddition

Org Biomol Chem. 2019 Mar 13;17(11):2892-2895. doi: 10.1039/c9ob00325h.

Abstract

The first organocatalytic method for the asymmetric construction of CF3-containing spiro-thiazolone-pyrrolidine compounds has been developed. This is one of the very few methods to reach spiro-thiazolones, and afforded the products in excellent yields and stereoselectivities catalysed by only 1 mol% cinchona alkaloid-derived catalyst.

Publication types

  • Research Support, Non-U.S. Gov't