De novo structure determination of 3-((3-aminopropyl)amino)-4-hydroxybenzoic acid, a novel and abundant metabolite in Acinetobacter baylyi ADP1

Metabolomics. 2019 Mar 14;15(3):45. doi: 10.1007/s11306-019-1508-3.

Abstract

Introduction: Metabolite identification remains a major bottleneck in the understanding of metabolism. Many metabolomics studies end up with unknown compounds, leaving a landscape of metabolites and metabolic pathways to be unraveled. Therefore, identifying novel compounds within a metabolome is an entry point into the 'dark side' of metabolism.

Objectives: This work aimed at elucidating the structure of a novel metabolite that was first detected in the soil bacterium Acinetobacter baylyi ADP1 (ADP1).

Methods: We used high resolution multi-stage tandem mass spectrometry for characterizing the metabolite within the metabolome. We purified the molecule for 1D- and 2D-NMR (1H, 13C, 1H-1H-COSY, 1H-13C-HSQC, 1H-13C-HMBC and 1H-15N-HMBC) analyses. Synthetic standards were chemically prepared from MS and NMR data interpretation.

Results: We determined the de novo structure of a previously unreported metabolite: 3-((3-aminopropyl)amino)-4-hydroxybenzoic acid. The proposed structure was validated by comparison to a synthetic standard. With a concentration in the millimolar range, this compound appears as a major metabolite in ADP1, which we anticipate to participate to an unsuspected metabolic pathway. This novel metabolite was also detected in another γ-proteobacterium.

Conclusion: Structure elucidation of this abundant and novel metabolite in ADP1 urges to decipher its biosynthetic pathway and cellular function.

Keywords: Bacterial metabolism; Functional genomics; LC/MS-Orbitrap; NMR; Structure elucidation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acinetobacter / chemistry
  • Acinetobacter / metabolism*
  • Magnetic Resonance Spectroscopy / methods
  • Metabolome
  • Metabolomics / methods
  • Parabens / chemistry*
  • Parabens / metabolism
  • Tandem Mass Spectrometry / methods

Substances

  • Parabens

Supplementary concepts

  • Acinetobacter baylyi