In Vitro Activity of Fenticonazole against Candida and Bacterial Vaginitis Isolates Determined by Mono- or Dual-Species Testing Assays

Antimicrob Agents Chemother. 2019 Jun 24;63(7):e02693-18. doi: 10.1128/AAC.02693-18. Print 2019 Jul.

Abstract

We determined the in vitro activity of fenticonazole against 318 vaginitis isolates of Candida and bacterial species and selected 28 isolates for time-kill studies. At concentrations equal to 4× MIC, fenticonazole reached the 99.9% killing endpoint by ∼10 h for Staphylococcus aureus, Streptococcus agalactiae, and Escherichia coli and by ∼17 h for Candida albicans and Candida parapsilosis; and at concentrations equal to 8× MIC, by ∼19 and ∼20 h for Candida glabrata and Candida tropicalis, respectively. At concentrations equal to 2× MIC, fenticonazole required ∼20 h to reach the above endpoint against C. albicans in mixed culture with S. aureus, S. agalactiae, or E. coli versus ∼17 h against C. albicans in pure culture. Supra-MICs are achievable in topically treated patients' vaginal surfaces.

Keywords: antimicrobial susceptibility testing; fenticonazole; targeted therapy; vaginal isolates.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / therapeutic use*
  • Antifungal Agents / therapeutic use*
  • Bacteria / drug effects*
  • Candida / drug effects*
  • Candidiasis / drug therapy*
  • Female
  • Humans
  • Imidazoles / therapeutic use*
  • Microbial Sensitivity Tests / methods
  • Vaginosis, Bacterial / drug therapy*

Substances

  • Anti-Bacterial Agents
  • Antifungal Agents
  • Imidazoles
  • fenticonazole