Light-Induced Redox-Responsive Smart Drug Delivery System by Using Selenium-Containing Polymer@MOF Shell/Core Nanocomposite

Adv Healthc Mater. 2019 Aug;8(15):e1900406. doi: 10.1002/adhm.201900406. Epub 2019 Jun 11.

Abstract

Rational design of controllable drug release systems is important for tumor treatments due to the nonspecific toxicity of many chemotherapeutics. Herein, laser or light responsive pharmaceutical delivery nanoparticles are designed, by taking the advantages of redox responsive selenium (Se) substituted polymer as shell and photosensitive porphyrin zirconium metal-organic frameworks (MOF) as core. In detail, redox cleavable di-(1-hydroxylundecyl) selenide (DH-Se), biocompatible poly(ethylene glycol) (PEG), and poly(propylene glycol) (PPG) are randomly polymerized to form poly(DH-Se/PEG/PPG urethane), which is used to coat the reactive oxygen species' (ROS) producible porous porphyrin zirconium metal organization formulation (PCN-224 MOF) to form the final poly(DH-Se/PEG/PPG urethane)@MOF shell-core nanoparticle with spherical shape by emulsion approach. Interestingly, poly(DH-Se/PEG/PPG urethane)@MOF nanoparticles with loading of chemotherapeutic doxorubicin (DOX) experience a fast and controllable release, which can realize the combination of chemotherapy and photodynamic therapy upon irradiation with laser light, due to the light-triggered ROS production by MOF which further causes the cleavage of poly(DH-Se/PEG/PPG urethane) polymer chain and the release of encapsulated DOX. To the best of the authors' knowledge, this is the first design of utilizing MOF and selenium substituted polymer as controllable drug release carriers, which might be beneficial for precise chemotherapy and photodynamic therapy combination.

Keywords: MOF; chemotherapy; drug delivery; photodynamic therapy; selenium.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibiotics, Antineoplastic / chemistry
  • Antibiotics, Antineoplastic / metabolism
  • Antibiotics, Antineoplastic / pharmacology
  • Antibiotics, Antineoplastic / therapeutic use
  • Cell Survival / drug effects
  • Doxorubicin / chemistry
  • Doxorubicin / metabolism
  • Doxorubicin / pharmacology
  • Doxorubicin / therapeutic use
  • Drug Carriers / chemistry*
  • Drug Liberation
  • Hep G2 Cells
  • Humans
  • Light*
  • Metal-Organic Frameworks / chemistry*
  • Mice
  • Mice, Nude
  • Nanocomposites / chemistry*
  • Neoplasms / drug therapy
  • Neoplasms / pathology
  • Neoplasms / therapy
  • Oxidation-Reduction
  • Polyethylene Glycols / chemistry
  • Polymers / chemistry*
  • Reactive Oxygen Species / metabolism
  • Selenium / chemistry*

Substances

  • Antibiotics, Antineoplastic
  • Drug Carriers
  • Metal-Organic Frameworks
  • Polymers
  • Reactive Oxygen Species
  • Polyethylene Glycols
  • Doxorubicin
  • Selenium