Effect of heat stress and Hsp90 inhibition on T-type calcium currents and voltage-dependent potassium currents in leydig cells

J Therm Biol. 2019 Aug:84:1-7. doi: 10.1016/j.jtherbio.2019.05.022. Epub 2019 May 23.

Abstract

Heat can trigger testicular damage and impair fertility. Leydig cells produce testosterone in response to stimulation by luteinizing hormone (LH), which induces Ca2+ entry and K+ efflux through ion channels in their plasma membrane. Considering that mechanisms coordinating the Leydig cell responses to hyperthermic stress remain unclear; the present study analyzed the effects of heat stress (HS, 43°C, 15 min) and inhibition of Hsp90 on T-type calcium currents and voltage-dependent potassium currents (VKC) in mice Leydig cells. Results show that HS reduced the VKC steady state currents at +80 mV (45.3%) and maximum conductance (71.5%), as well as increased the activation time constant (31.7%) and the voltage for which half the channels are open (30%). Hsp90 inhibition did not change the VKC currents. T-type calcium currents were not affected by HS or Hsp90 inhibition. In conclusion, HS can slow the activation, reduce the currents and voltage dependence of the VKC, suggesting a possible role of these currents in the response to hyperthermic stress in Leydig cells.

Keywords: Calcium currents; High temperature; Hsp90; Ion channels; Leydig cells; Potassium currents.

MeSH terms

  • Animals
  • Benzoquinones / pharmacology
  • Calcium Channels, T-Type / physiology*
  • HSP90 Heat-Shock Proteins / antagonists & inhibitors
  • HSP90 Heat-Shock Proteins / physiology*
  • Heat-Shock Response / physiology*
  • Hot Temperature
  • Lactams, Macrocyclic / pharmacology
  • Leydig Cells / drug effects
  • Leydig Cells / physiology*
  • Male
  • Mice
  • Potassium Channels, Voltage-Gated / physiology*

Substances

  • 17-(3'-(dimethylamino)-1'-propyl)amino-17-demethoxygeldanamycin
  • Benzoquinones
  • Calcium Channels, T-Type
  • HSP90 Heat-Shock Proteins
  • Lactams, Macrocyclic
  • Potassium Channels, Voltage-Gated