Experimental and investigational drugs for the treatment of alpha-1 antitrypsin deficiency

Expert Opin Investig Drugs. 2019 Oct;28(10):891-902. doi: 10.1080/13543784.2019.1672656. Epub 2019 Oct 11.

Abstract

Introduction: Alpha-1 antitrypsin deficiency (AATD) is most often associated with chronic lung disease, early onset emphysema, and liver disease. The standard of care in lung disease due to AATD is alpha-1 antitrypsin augmentation but there are several new and emerging treatment options under investigation for both lung and liver manifestations. Areas covered: We review therapeutic approaches to lung and liver disease in alpha-1 antitrypsin deficiency (AATD) and the agents in clinical development according to their mode of action. The focus is on products in clinical trials, but data from pre-clinical studies are described where relevant, particularly where progression to trials appears likely. Expert opinion: Clinical trials directed at lung and liver disease separately are now taking place. Multimodality treatment may be the future, but this could be limited by treatment costs. The next 5-10 years may reveal new guidance on when to use therapeutics for slowing disease progression with personalized treatment regimes coming to the forefront.

Keywords: Alpha-1 antitrypsin deficiency; chronic obstructive pulmonary disease; cirrhosis; clinical trials; emphysema.

Publication types

  • Review

MeSH terms

  • Animals
  • Disease Progression
  • Drug Development / methods*
  • Drugs, Investigational / administration & dosage*
  • Drugs, Investigational / pharmacology
  • Humans
  • Liver Diseases / drug therapy
  • Liver Diseases / etiology
  • Lung Diseases / drug therapy
  • Lung Diseases / etiology
  • Precision Medicine / methods
  • alpha 1-Antitrypsin Deficiency / drug therapy*
  • alpha 1-Antitrypsin Deficiency / physiopathology

Substances

  • Drugs, Investigational