Disease-associated mutations in Niemann-Pick type C1 alter ER calcium signaling and neuronal plasticity

J Cell Biol. 2019 Dec 2;218(12):4141-4156. doi: 10.1083/jcb.201903018. Epub 2019 Oct 10.

Abstract

Niemann-Pick type C1 (NPC1) protein is essential for the transport of externally derived cholesterol from lysosomes to other organelles. Deficiency of NPC1 underlies the progressive NPC1 neurodegenerative disorder. Currently, there are no curative therapies for this fatal disease. Given the Ca2+ hypothesis of neurodegeneration, which posits that altered Ca2+ dynamics contribute to neuropathology, we tested if disease mutations in NPC1 alter Ca2+ signaling and neuronal plasticity. We determine that NPC1 inhibition or disease mutations potentiate store-operated Ca2+ entry (SOCE) due to a presenilin 1 (PSEN1)-dependent reduction in ER Ca2+ levels alongside elevated expression of the molecular SOCE components ORAI1 and STIM1. Associated with this dysfunctional Ca2+ signaling is destabilization of neuronal dendritic spines. Knockdown of PSEN1 or inhibition of the SREBP pathway restores Ca2+ homeostasis, corrects differential protein expression, reduces cholesterol accumulation, and rescues spine density. These findings highlight lysosomes as a crucial signaling platform responsible for tuning ER Ca2+ signaling, SOCE, and synaptic architecture in health and disease.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium Signaling*
  • Carrier Proteins / metabolism
  • Cholesterol / metabolism
  • Dendritic Spines / metabolism
  • Endoplasmic Reticulum / metabolism*
  • Fibroblasts / metabolism
  • Hippocampus / cytology
  • Humans
  • Intracellular Signaling Peptides and Proteins / genetics
  • Intracellular Signaling Peptides and Proteins / metabolism*
  • Lysosomes / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mutation
  • Neoplasm Proteins / metabolism
  • Neurodegenerative Diseases / metabolism
  • Neuronal Plasticity*
  • Neurons / metabolism
  • Niemann-Pick C1 Protein
  • ORAI1 Protein / metabolism
  • Presenilin-1 / metabolism
  • Signal Transduction
  • Stromal Interaction Molecule 1 / metabolism
  • Synapses / metabolism

Substances

  • Carrier Proteins
  • Intracellular Signaling Peptides and Proteins
  • NPC1 protein, human
  • Neoplasm Proteins
  • Niemann-Pick C1 Protein
  • ORAI1 Protein
  • ORAI1 protein, human
  • PSEN1 protein, human
  • Presenilin-1
  • STIM1 protein, human
  • Stromal Interaction Molecule 1
  • Cholesterol