In vitro activity of meropenem/piperacillin/tazobactam triple combination therapy against clinical isolates of Staphylococcus aureus, Staphylococcus epidermidis, Staphylococcus pseudintermedius and vancomycin-resistant Enterococcus spp

Int J Antimicrob Agents. 2020 Feb;55(2):105864. doi: 10.1016/j.ijantimicag.2019.105864. Epub 2019 Dec 20.

Abstract

Objectives: To evaluate the activity of the reported synergistic and collaterally sensitive antibiotic combination, meropenem/piperacillin/tazobactam (ME/PI/TZ), against a panel of methicillin-resistant Staphylococcus aureus (MRSA) and other methicillin-resistant Staphylococcus species; and to investigate the relationship between ME/PI/TZ susceptibility and the genomic background of clinical isolates of MRSA.

Methods: ME/PI/TZ combination and single drug minimum inhibitory concentrations (MICs) were determined for 207 strains (including 121 MRSA, 4 methicillin-sensitive S. aureus [MSSA], 37 vancomycin-intermediate S. aureus [VISA], 6 ceftaroline non-susceptible MRSA, 29 coagulase-negative staphylococci [CoNS], 5 S. pseudointermedius and 5 vancomycin-resistant Enterococci [VRE]) by broth microdilution. Whole genomes of 168 S. aureus strains were sequenced, assembled, and comparatively analysed.

Results: USA300-SCCmec type IV isolates, clonal complex 8 (CC8)-MRSA isolates, including some VISA and ceftaroline (CPT)-intermediate strains, and all tested methicillin-resistant S. epidermidis isolates were highly susceptible to ME/PI/TZ. Isolates with elevated MICs (MICs of >16/16/16 mg/L) clustered with the USA100-SCCmec type II strain. Susceptibility of MRSA to ME/PI/TZ was correlated with susceptibility to ME. No obvious cross-resistance to CPT was observed among high-ME/PI/TZ MIC isolates.

Conclusions: The ME/PI/TZ combination is effective against a variety of clinical MRSA isolates, particularly of the USA300 lineage, which is expanding worldwide. ME/PI/TZ is also effective against drug-resistant CoNS and S. pseudintermedius clinical isolates.

Keywords: Antibiotic combination; Antibiotic resistance; Clinical isolates; MRSA; Staphylococci; Whole-genome sequencing.

MeSH terms

  • Anti-Bacterial Agents / therapeutic use*
  • Drug Resistance, Multiple, Bacterial / genetics
  • Drug Therapy, Combination
  • Genome, Bacterial / genetics
  • Genomics
  • Humans
  • Meropenem / therapeutic use*
  • Methicillin-Resistant Staphylococcus aureus / drug effects
  • Methicillin-Resistant Staphylococcus aureus / genetics
  • Microbial Sensitivity Tests
  • Piperacillin / therapeutic use*
  • Staphylococcal Infections / drug therapy*
  • Staphylococcus / drug effects
  • Staphylococcus / genetics
  • Staphylococcus epidermidis / drug effects
  • Staphylococcus epidermidis / genetics
  • Tazobactam / therapeutic use*
  • Vancomycin-Resistant Enterococci / drug effects*
  • Vancomycin-Resistant Enterococci / genetics
  • Whole Genome Sequencing
  • beta-Lactamase Inhibitors / therapeutic use

Substances

  • Anti-Bacterial Agents
  • beta-Lactamase Inhibitors
  • Meropenem
  • Tazobactam
  • Piperacillin

Supplementary concepts

  • Staphylococcus pseudintermedius