Antibody Opsonization of a TLR9 Agonist-Containing Virus-like Particle Enhances In Situ Immunization

J Immunol. 2020 Mar 1;204(5):1386-1394. doi: 10.4049/jimmunol.1900742. Epub 2020 Jan 17.

Abstract

The immunologic and therapeutic effects of intratumoral (IT) delivery of a novel virus-like particle as a lymphoma immunotherapy were evaluated in preclinical studies with human cells and a murine model. CMP-001 is a virus-like particle composed of the Qβ bacteriophage capsid protein encapsulating an immunostimulatory CpG-A oligodeoxynucleotide TLR9 agonist. In vitro, CMP-001 induced cytokine production, including IFN-α from plasmacytoid dendritic cells, but only in the presence of anti-Qβ Ab. In vivo, IT CMP-001 treatment of murine A20 lymphoma enhanced survival and reduced growth of both injected and contralateral noninjected tumors in a manner dependent on both the ability of mice to generate anti-Qβ Ab and the presence of T cells. The combination of IT CMP-001 with systemic anti-PD-1 enhanced antitumor responses in both injected and noninjected tumors. IT CMP-001 alone or combined with anti-PD-1 augmented T cell infiltration in tumor-draining lymph nodes. We conclude IT CMP-001 induces a robust antitumor T cell response in an anti-Qβ Ab-dependent manner and results in systemic antitumor T cell effects that are enhanced by anti-PD-1 in a mouse model of B cell lymphoma. Early-phase clinical evaluation of CMP-001 and anti-PD-1 combination therapy in lymphoma will begin shortly, based in part on these results.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies, Neoplasm / immunology
  • Cell Line, Tumor
  • Female
  • Humans
  • Immunity, Cellular / drug effects*
  • Immunization*
  • Lymphoma* / immunology
  • Lymphoma* / pathology
  • Lymphoma* / therapy
  • Mice
  • Mice, Knockout
  • Oligodeoxyribonucleotides / pharmacology*
  • Toll-Like Receptor 9* / agonists
  • Toll-Like Receptor 9* / immunology
  • Vaccines, Virus-Like Particle / pharmacology*

Substances

  • Antibodies, Neoplasm
  • CPG-oligonucleotide
  • Oligodeoxyribonucleotides
  • Tlr9 protein, mouse
  • Toll-Like Receptor 9
  • Vaccines, Virus-Like Particle