Cytotoxicity, sister-chromatid exchange, chromosome aberration and transformation induced by 2,2-dichlorovinyl-O,O-dimethyl phosphate

Mutat Res. 1988 Dec;206(4):439-45. doi: 10.1016/0165-1218(88)90051-1.

Abstract

2,2-Dichlorovinyl-O,O-dimethyl phosphate (DDVP), an extensively used household insecticide, was assayed for its genotoxicity in primary rat tracheal epithelial (RTE) cells. Cytotoxicity of DDVP to RTE cells was dose-dependent, killing about 50% of the cell population at a dose of 80 micrograms/ml. Sister-chromatid exchange (SCE) and chromosomal aberrations induced by this insecticide were positive in RTE cells although the doses needed for significant inductions were much higher than those by a known genotoxic agent, N-methyl-N'-nitro-N-nitrosoguanidine (MNNG). The level of transformation induced by DDVP in RTE cells was about 1/5 that induced by MNNG at a dose of similar cytotoxicity. The slope of the regression line for induced transformation is 1.27. DDVP probably induces the genotoxic effect in RTE cells by a one-hit mechanism.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Survival / drug effects
  • Cell Transformation, Neoplastic / chemically induced*
  • Cells, Cultured
  • Chromosome Aberrations*
  • Dichlorvos / pharmacology*
  • Epithelium / drug effects
  • Male
  • Methylnitronitrosoguanidine / pharmacology
  • Mutagenicity Tests
  • Rats
  • Rats, Inbred Strains
  • Sister Chromatid Exchange / drug effects*
  • Trachea

Substances

  • Methylnitronitrosoguanidine
  • Dichlorvos