Changes in Renal Function After Switching From TDF to TAF in HIV-Infected Individuals: A Prospective Cohort Study

J Infect Dis. 2020 Jul 23;222(4):637-645. doi: 10.1093/infdis/jiaa125.

Abstract

Background: Replacing tenofovir disoproxil fumarate (TDF) with tenofovir alafenamide (TAF) improves renal tubular markers in HIV-infected individuals but the impact on estimated glomerular filtration rate (eGFR) remains unclear.

Methods: In all participants from the Swiss HIV Cohort Study who switched from TDF to TAF-containing antiretroviral regimen or continued TDF, we estimated changes in eGFR and urine protein-to-creatinine ratio (UPCR) after 18 months using mixed-effect models.

Results: Of 3520 participants (26.6% women, median age 50 years), 2404 (68.5%) switched to TAF. Overall, 1664 (47.3%) had an eGFR <90 mL/min and 1087 (30.9%) an UPCR ≥15 mg/mmol. In patients with baseline eGFR ≥90 mL/min, eGFR decreased with the use of TDF and TAF (-1.7 mL/min). Switching to TAF was associated with increases in eGFR of 1.5 mL/min (95% confidence interval [CI], .5-2.5) if the baseline eGFR was 60-89 mL/min, and 4.1 mL/min (95% CI, 1.6-6.6) if <60 mL/min. In contrast, eGFR decreased by 5.8 mL/min (95% CI, 2.3-9.3) with continued use of TDF in individuals with baseline eGFR <60 mL/min. UPCR decreased after replacing TDF by TAF, independent of baseline eGFR.

Conclusions: Switching from TDF to TAF improves eGFR and proteinuria in patients with renal dysfunction.

Keywords: antiretroviral therapy; comorbidities; estimated glomerular filtration rate; renal tubulopathy; switch; tenofovir alafenamide; urine protein-to-creatinine ratio.

Publication types

  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / therapeutic use
  • Adult
  • Alanine
  • Anti-HIV Agents / therapeutic use*
  • Drug Substitution*
  • Female
  • Glomerular Filtration Rate*
  • HIV Infections / drug therapy*
  • Humans
  • Kidney Function Tests
  • Male
  • Middle Aged
  • Prospective Studies
  • Switzerland
  • Tenofovir / therapeutic use*

Substances

  • Anti-HIV Agents
  • Tenofovir
  • tenofovir alafenamide
  • Adenine
  • Alanine