Cartilage repair mediated by thermosensitive photocrosslinkable TGFβ1-loaded GM-HPCH via immunomodulating macrophages, recruiting MSCs and promoting chondrogenesis

Theranostics. 2020 Feb 3;10(6):2872-2887. doi: 10.7150/thno.41622. eCollection 2020.

Abstract

Repairing cartilage defects using thermosensitive hydrogels is an attractive treatment strategy, but the poor mechanical properties and limited understanding of the interactions between hydrogels and cells limit their application. Methods: In this study, a thermosensitive hydroxypropyl chitin hydrogel (HPCH) was functionalized with methacrylate groups to synthesize photocrosslinkable glycidyl methacrylate-modified HPCH (GM-HPCH). GM-HPCH could form a gel in situ through a thermosensitive sol-gel transition and its mechanical properties can be improved by UV irradiation. Cell viability, cell adhesion and anti-apoptosis activity of GM-HPCH were evaluated. Transforming growth factor-β1 (TGFβ1) was introduced into the GM-HPCH hydrogel to fabricate the composite hydrogel. The macrophage immunomodulation, MSC recruitment and chondrogenesis of the composite hydrogel were evaluated. Results: With high biocompatibility, GM-HPCH could protect chondrocytes from apoptosis. Both the in vitro and in vivo experiments showed that GM-HPCH + TGFβ1 shifted the recruited macrophages from M1 to M2 and promoted chondrogenic gene expression. Additionally, the composite hydrogel could promote the migration of marrow stromal cells (MSCs) in the Transwell test and increase migrated gene expression. The fluorescent tracking of MSCs confirmed MSC homing in the rat chondral defect with the help of GM-HPCH. The macroscopic evaluation and histological results at 6 weeks and 12 weeks postsurgery showed that GM-HPCH + TGFβ1 can achieve superior cartilage healing. Conclusions: The GM-HPCH + TGFβ1 hydrogel effectively promoted cartilage repair via immunomodulating macrophages, recruiting MSCs and promoting chondrogenesis; thus it is a promising injectable hydrogel for cartilage regeneration.

Keywords: TGFβ1; cartilage tissue engineering; cell recruitment; immunomodulation; mechanical improvement; thermosensitive photocrosslinkable hydrogel.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cartilage Diseases / therapy*
  • Cell Adhesion / drug effects
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Cell- and Tissue-Based Therapy
  • Chitin / analogs & derivatives
  • Chitin / pharmacology*
  • Chondrogenesis / drug effects*
  • Human Umbilical Vein Endothelial Cells
  • Humans
  • Hydrogels* / pharmacology
  • Hydrogels* / therapeutic use
  • Male
  • Mesenchymal Stem Cells
  • Mice
  • RAW 264.7 Cells
  • Rats
  • Rats, Sprague-Dawley
  • Tissue Engineering
  • Transforming Growth Factor beta1 / pharmacology*
  • Transforming Growth Factor beta1 / therapeutic use

Substances

  • Hydrogels
  • Transforming Growth Factor beta1
  • Chitin