Metformin Enhances the Antitumor Activity of CD8+ T Lymphocytes via the AMPK-miR-107-Eomes-PD-1 Pathway

J Immunol. 2020 May 1;204(9):2575-2588. doi: 10.4049/jimmunol.1901213. Epub 2020 Mar 27.

Abstract

Metformin has been studied for its anticancer effects by regulating T cell functions. However, the mechanisms through which metformin stimulates the differentiation of memory T cells remain unclear. We found that the frequencies of memory stem and central memory T cells increased for both in peripheral and tumor-infiltrating CD8+ T cells in metformin-treated lung cancer patients compared with those not taking the medication. An in vitro assay showed that metformin promoted the formation of memory CD8+ T cells and enhanced their antiapoptotic abilities. In addition, AMP-activated protein kinase (AMPK) activation decreased microRNA-107 expression, thus enhancing Eomesodermin expression, which suppressed the transcription of PDCD1 in metformin-treated CD8+ T cells. In the CAR-T cell therapy model, metformin also exhibited cytotoxicity-promoting effects that led to decreased tumor growth. Metformin could reprogram the differentiation of CD8+ T cells, which may benefit the clinical therapy of cancer patients by facilitating long-lasting cytotoxic functions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • A549 Cells
  • AMP-Activated Protein Kinases / metabolism*
  • Antineoplastic Agents / metabolism*
  • Apoptosis / drug effects
  • CD8-Positive T-Lymphocytes / drug effects*
  • CD8-Positive T-Lymphocytes / metabolism
  • Cell Differentiation / drug effects
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • HCT116 Cells
  • Humans
  • Immunologic Memory / drug effects
  • Metformin / pharmacology*
  • MicroRNAs / metabolism*
  • Programmed Cell Death 1 Receptor / metabolism*
  • Retrospective Studies
  • Signal Transduction / drug effects
  • T-Box Domain Proteins / metabolism*
  • Transcription, Genetic / drug effects

Substances

  • Antineoplastic Agents
  • EOMES protein, human
  • MIRN107 microRNA, human
  • MicroRNAs
  • PDCD1 protein, human
  • Programmed Cell Death 1 Receptor
  • T-Box Domain Proteins
  • Metformin
  • AMP-Activated Protein Kinases