A mitochondria-targeting NIR fluorescent potassium ion sensor: real-time investigation of the mitochondrial K+ regulation of apoptosis in situ

Chem Commun (Camb). 2020 May 19;56(40):5405-5408. doi: 10.1039/d0cc00579g.

Abstract

The first NIR fluorescent mitochondria-targeting K+ sensor, denoted as TAC-Rh, was developed. The produced sensor consists of a rhodamine analog as the fluorophore and triazacryptand (TAC) as the K+ recognition unit. Compared to the K+ sensors reported previously, TAC-Rh exhibits two unique optical properties: the largest Stokes shifts (120 nm) and the longest emission peak wavelength (720 nm). With the assistance of this novel sensor, real-time changes of K+ concentrations in mitochondria during apoptosis were monitored for the first time. Moreover, it was also the first time that the relationship between mitochondrial K+ flux and apoptosis was investigated in real time using fluorescence imaging.

MeSH terms

  • Apoptosis / physiology*
  • Azabicyclo Compounds / chemistry
  • Cell Line, Tumor
  • Fluorescent Dyes / chemistry*
  • Humans
  • Microscopy, Confocal / methods
  • Microscopy, Fluorescence / methods
  • Mitochondria / metabolism*
  • Potassium / analysis*
  • Potassium / metabolism
  • Rhodamines / chemistry

Substances

  • 1,4,7,10,13,16,21,24-octaazabicyclo(8.8.8)hexacosane
  • Azabicyclo Compounds
  • Fluorescent Dyes
  • Rhodamines
  • Potassium