Epoxy-Tethered Diels-Alder Reaction toward the Tricyclic Core of Kalihinols

Org Lett. 2020 May 1;22(9):3557-3560. doi: 10.1021/acs.orglett.0c00998. Epub 2020 Apr 15.

Abstract

A chiral-template-driven intramolecular Diels-Alder reaction has been used to build the tricyclic core of kalihinols, a group of antimalarial marine natural products. The key starting materials are commercially available nerol and sulcatone.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biological Products*
  • Cycloaddition Reaction
  • Molecular Structure

Substances

  • Biological Products