A conformation-based intra-molecular initiation factor identified in the flavivirus RNA-dependent RNA polymerase

PLoS Pathog. 2020 May 1;16(5):e1008484. doi: 10.1371/journal.ppat.1008484. eCollection 2020 May.

Abstract

The flaviviruses pose serious threats to human health. Being a natural fusion of a methyltransferase (MTase) and an RNA-dependent RNA polymerase (RdRP), NS5 is the most conserved flavivirus protein and an important antiviral target. Previously reported NS5 structures represented by those from the Japanese encephalitis virus (JEV) and Dengue virus serotype 3 (DENV3) exhibit two apparently different global conformations, defining two sets of intra-molecular MTase-RdRP interactions. However, whether these NS5 conformations are conserved in flaviviruses and their specific functions remain elusive. Here we report two forms of DENV serotype 2 (DENV2) NS5 crystal structures representing two conformational states with defined analogies to the JEV-mode and DENV3-mode conformations, respectively, demonstrating the conservation of both conformation modes and providing clues for how different conformational states may be interconnected. Data from in vitro polymerase assays further demonstrate that perturbing the JEV-mode but not the DENV3-mode intra-molecular interactions inhibits catalysis only at initiation, while the cell-based virological analysis suggests that both modes of interactions are important for virus proliferation. Our work highlights the role of MTase as a unique intra-molecular initiation factor specifically only through the JEV-mode conformation, providing an example of conformation-based crosstalk between naturally fused protein functional modules.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cricetinae
  • Crystallography, X-Ray
  • Dengue Virus / chemistry*
  • Dengue Virus / metabolism
  • Encephalitis Virus, Japanese / chemistry*
  • Encephalitis Virus, Japanese / metabolism
  • Humans
  • Protein Domains
  • RNA-Dependent RNA Polymerase / chemistry*
  • RNA-Dependent RNA Polymerase / metabolism
  • Viral Nonstructural Proteins / chemistry*
  • Viral Nonstructural Proteins / metabolism

Substances

  • NS5 protein, dengue virus
  • NS5 protein, flavivirus
  • Viral Nonstructural Proteins
  • RNA-Dependent RNA Polymerase

Grants and funding

This work was supported by the National Key Research and Development Program of China (www.most.gov.cn, 2018YFA0507200 to PG, and 2016YFC1200400 to HQY), the National Natural Science Foundation of China (www.nsfc.gov.cn, 31670154 to PG and 31370198 to PG).The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.