Randomized controlled trial of landiolol, a short-acting beta-1 adrenergic receptor blocker, illustrating changes in high-molecular weight adiponectin levels after elective percutaneous coronary intervention

Heart Vessels. 2020 Nov;35(11):1510-1517. doi: 10.1007/s00380-020-01637-6. Epub 2020 Jun 12.

Abstract

Adiponectin (APN) has cardioprotective properties and bisoprolol has been reported to increase myocardial APN expression and reduce myocardial damage. Administration of landiolol, which has a higher cardio-selectivity and shorter half-life than bisoprolol, during the percutaneous coronary intervention (PCI) may increase serum APN and high-molecular weight (HMW)-APN, an active form of APN, in patients with stable angina pectoris (SAP). We recruited 70 patients with SAP and randomized them to intravenous landiolol during PCI (N = 35) or control group (N = 35). The primary endpoint was serum APN and HMW-APN level 3 days after PCI. There was no difference in the primary endpoint between the landiolol and control groups (8.93 ± 5.24 vs. 10.18 ± 5.81 μg/mL, p = 0.35 and 3.36 ± 2.75 vs. 4.28 ± 3.13 μg/mL, p = 0.20) for APN and HMW-APN levels, respectively. APN and HMW-APN level were significantly decreased 1 day after PCI [-0.55 ± 0.92 μg/mL (9.87-9.32 μg/mL), p < 0.001 and -0.20 ± 0.45 μg/mL (3.89-3.69 μg/mL), p < 0.001, respectively]. Additionally, the absolute change in HMW-APN was significantly smaller in the landiolol group compared to the control group (-0.08 ± 0.27 vs. -0.31 ± 0.55 μg/mL, p = 0.031). Multiple linear regression analysis showed that use of landiolol was an independent predictor of change in HMW-APN (β = 0.276, p = 0.014). Serum APN and HMW-APN level 3 days after PCI were similar between patients treated with and without landiolol. APN and HMW-APN decreased 1 day after PCI in the SAP and landiolol mitigated decrease in HMW-APN.

Keywords: Adiponectin; Adrenergic beta-antagonist; Coronary artery disease; Landiolol; Percutaneous coronary intervention.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Adiponectin / blood*
  • Adrenergic beta-1 Receptor Antagonists / administration & dosage*
  • Adrenergic beta-1 Receptor Antagonists / adverse effects
  • Aged
  • Aged, 80 and over
  • Angina, Stable / blood
  • Angina, Stable / diagnosis
  • Angina, Stable / therapy*
  • Biomarkers / blood
  • Coronary Artery Disease / blood
  • Coronary Artery Disease / diagnostic imaging
  • Coronary Artery Disease / therapy*
  • Female
  • Humans
  • Japan
  • Male
  • Middle Aged
  • Molecular Weight
  • Morpholines / administration & dosage*
  • Morpholines / adverse effects
  • Percutaneous Coronary Intervention* / adverse effects
  • Prospective Studies
  • Time Factors
  • Treatment Outcome
  • Urea / administration & dosage
  • Urea / adverse effects
  • Urea / analogs & derivatives*

Substances

  • ADIPOQ protein, human
  • Adiponectin
  • Adrenergic beta-1 Receptor Antagonists
  • Biomarkers
  • Morpholines
  • landiolol
  • Urea