Abstract
Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is responsible for millions of infections and hundreds of thousands of deaths globally. There are no widely available licensed therapeutics against SARS-CoV-2, highlighting an urgent need for effective interventions. The virus enters host cells through binding of a receptor-binding domain within its trimeric spike glycoprotein to human angiotensin-converting enzyme 2. In this article, we describe the generation and characterization of a panel of murine mAbs directed against the receptor-binding domain. One mAb, 2B04, neutralized wild-type SARS-CoV-2 in vitro with remarkable potency (half-maximal inhibitory concentration of <2 ng/ml). In a murine model of SARS-CoV-2 infection, 2B04 protected challenged animals from weight loss, reduced lung viral load, and blocked systemic dissemination. Thus, 2B04 is a promising candidate for an effective antiviral that can be used to prevent SARS-CoV-2 infection.
Copyright © 2020 by The American Association of Immunologists, Inc.
Publication types
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Research Support, N.I.H., Extramural
MeSH terms
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Angiotensin-Converting Enzyme 2
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Animals
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Antibodies, Monoclonal / immunology
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Antibodies, Monoclonal / pharmacology
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Antibodies, Monoclonal / therapeutic use*
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Antibodies, Neutralizing / immunology
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Antibodies, Neutralizing / pharmacology
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Antibodies, Neutralizing / therapeutic use*
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Antibodies, Viral / immunology
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Antibodies, Viral / pharmacology
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Antibodies, Viral / therapeutic use*
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Betacoronavirus / drug effects*
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COVID-19
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Chlorocebus aethiops
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Coronavirus Infections / drug therapy*
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Coronavirus Infections / immunology*
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Coronavirus Infections / virology
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Disease Models, Animal
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Epitope Mapping
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Female
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HEK293 Cells
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Humans
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Immunodominant Epitopes / immunology
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Mice
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Mice, Inbred C57BL
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Pandemics
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Peptidyl-Dipeptidase A / genetics
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Peptidyl-Dipeptidase A / metabolism
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Pneumonia, Viral / drug therapy*
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Pneumonia, Viral / immunology*
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Pneumonia, Viral / virology
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Protein Interaction Domains and Motifs / genetics
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Protein Interaction Domains and Motifs / immunology
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SARS-CoV-2
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Spike Glycoprotein, Coronavirus / chemistry
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Spike Glycoprotein, Coronavirus / metabolism
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Transfection
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Vero Cells
Substances
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Antibodies, Monoclonal
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Antibodies, Neutralizing
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Antibodies, Viral
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Immunodominant Epitopes
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Spike Glycoprotein, Coronavirus
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spike protein, SARS-CoV-2
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Peptidyl-Dipeptidase A
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ACE2 protein, human
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Ace2 protein, mouse
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Angiotensin-Converting Enzyme 2